SCHEMBL2397615

SCHEMBL2397615

CC(C)(C)c1ncc(-c2ccc3nc(Nc4cccc(N[C@H]5CC[C@H](O)CC5)n4)sc3n2)cc1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITK Q08881 6/20 0.39
LCK P06239 4/20 0.39
AURKB Q96GD4 3/20 0.39
MAPK8 P45983 2/20 0.37
MAPK9 P45984 2/20 0.37
HSP90AA1 P07900 8/20 0.36
MELK Q14680 1/20 0.35
CCNT1 O60563 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2397725 0.78 ITK (0.50) ITKLCKAURKBCCNT1
SCHEMBL2397731 0.78 ITK (0.50) ITKLCKAURKBCCNT1
SCHEMBL2396989 0.77 PIK3CG (0.49) ITKLCKAURKBHSP90AA1
SCHEMBL2396976 0.77 PIK3CG (0.49) ITKLCKAURKBHSP90AA1
Trifluoroacetic Acid SCHEMBL2370610 0.77 IRAK4 (0.41) ITKLCKAURKBMAPK8MELK
SCHEMBL2395099 0.76 ITK (0.43) ITKLCKAURKBMELKCCNT1
SCHEMBL2395088 0.76 ITK (0.43) ITKLCKAURKBMELKCCNT1
SCHEMBL2396521 0.74 DYRK1A (0.41) ITKLCKAURKBCCNT1
SCHEMBL2370861 0.72 ITK (0.49) ITKLCKAURKBCCNT1
SCHEMBL2370869 0.72 ITK (0.49) ITKLCKAURKBCCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011110575-A1 DERIVATIVES OF 2-[2-(BENZO- OR PYRIDO-) THIAZOLYLAMINO]-6-AMINOPYRIDINE, USEFUL IN THE TREATMENT OF RESPIRATORIC, ALLERGIC OR INFLAMMATORY DISEASES GLAXO GROUP LIMITED (GB) 2011-09-15 WO disclosed