SCHEMBL23978126

SCHEMBL23978126

C=C(I)c1ccc(C)cc1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.44
TP53 P04637 1/20 0.44
NFE2L2 Q16236 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
KMT2A Q03164 2/20 0.39
HTT P42858 1/20 0.39
HSD11B1 P28845 1/20 0.38
FLT1 P17948 1/20 0.36
FLT4 P35916 1/20 0.36
KDR P35968 1/20 0.36
TRPA1 O75762 1/20 0.36
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2A6 P11509 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6547363 0.81 TDP1 (0.48) TDP1TP53NFE2L2SMN1; SMN2KMT2A
SCHEMBL753384 0.81 TDP1 (0.48) TDP1TP53NFE2L2SMN1; SMN2KMT2A
SCHEMBL29883022 0.81 TDP1 (0.48) TDP1TP53NFE2L2SMN1; SMN2KMT2A
SCHEMBL674175 0.79 TDP1 (0.46) TDP1TP53NFE2L2SMN1; SMN2KMT2A
SCHEMBL29444190 0.79 TDP1 (0.46) TDP1TP53NFE2L2SMN1; SMN2KMT2A
SCHEMBL11300977 0.79 TDP1 (0.46) TDP1TP53NFE2L2SMN1; SMN2KMT2A
SCHEMBL19908690 0.77 TDP1 (0.44) TDP1TP53NFE2L2SMN1; SMN2KMT2A
SCHEMBL6113079 0.77 NFE2L2 (0.47) TDP1TP53NFE2L2SMN1; SMN2KMT2A
SCHEMBL11601038 0.77 TDP1 (0.44) TDP1TP53NFE2L2SMN1; SMN2KMT2A
SCHEMBL11829383 0.77 SMN1; SMN2 (0.42) TDP1TP53NFE2L2SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021219578-A1 ANTIBACTERIAL 8-PHENYLAMINO-3-(PYRAZOL-4-YL)IMIDAZO[1,2-A]PYRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2021-11-04 WO disclosed