SCHEMBL23978696

SCHEMBL23978696

NC(=O)NC[C@H](NC(=O)c1c(Cl)cc(C(=O)NCc2cccc(Cl)c2)cc1Cl)C(=O)OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.46
NPC1 O15118 5/20 0.43
RAB9A P51151 4/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
ALDH1A1 P00352 2/20 0.42
TP53 P04637 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
HCRTR1 O43613 1/20 0.41
POLB P06746 3/20 0.40
MAPT P10636 3/20 0.40
CXCR3 P49682 1/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
APEX1 P27695 1/20 0.40
ALOX12 P18054 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23979010 0.90 NPC1 (0.42) NPC1SMN1; SMN2MEN1KMT2AHCRTR1
SCHEMBL23979030 0.89 NPC1 (0.46) NPC1MEN1KMT2AHCRTR1APEX1
SCHEMBL23978995 0.86 TACR1 (0.42) TACR1NPC1RAB9ACYP1A2CYP2D6
SCHEMBL26502639 0.86 TACR1 (0.42) TACR1NPC1RAB9ACYP1A2CYP2D6
SCHEMBL23978829 0.85 ITGB1 (0.46) TACR1NPC1ALDH1A1TP53MEN1
SCHEMBL23978850 0.84 KDM4E (0.42) TACR1SMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL24803383 0.82 EPHX2 (0.42) TACR1
SCHEMBL30083842 0.82 EPHX2 (0.42) TACR1
SCHEMBL26498658 0.82 EPHX2 (0.42) TACR1
SCHEMBL26508696 0.82 TRPV1 (0.43) TACR1NPC1RAB9ACYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed