SCHEMBL23979140

SCHEMBL23979140

C=C(CC)c1c(Cl)cc(C(=O)NCc2ccc(Cl)c(Cl)c2)cc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.54
LMNA P02545 1/20 0.54
HDAC4 P56524 1/20 0.53
HDAC1 Q13547 1/20 0.53
HDAC7 Q8WUI4 1/20 0.53
HDAC11 Q96DB2 1/20 0.53
HDAC8 Q9BY41 1/20 0.53
HDAC6 Q9UBN7 1/20 0.53
HDAC9 Q9UKV0 1/20 0.53
HDAC5 Q9UQL6 1/20 0.53
TSHR P16473 2/20 0.52
HPGD P15428 2/20 0.52
SMN1; SMN2 Q16637 1/20 0.51
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
KMT2A Q03164 1/20 0.49
MAOB P27338 1/20 0.47
WDR5 P61964 3/20 0.47
CCR2 P41597 1/20 0.46
APEX1 P27695 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23979113 0.87 EPHX2 (0.57) EPHX2LMNAHDAC4HDAC1HDAC7
SCHEMBL23979143 0.84 EPHX2 (0.59) EPHX2LMNAHDAC4HDAC1HDAC7
SCHEMBL23978806 0.82 EPHX2 (0.69) EPHX2LMNAHDAC4HDAC1HDAC7
SCHEMBL23979111 0.82 LMNA (0.63) EPHX2LMNAHDAC4HDAC1HDAC7
SCHEMBL8108036 0.80 EPHX2 (0.79) EPHX2LMNAHDAC4HDAC1HDAC7
SCHEMBL23978777 0.80 ROCK2 (0.48) MEN1KMT2A
SCHEMBL13026611 0.78 LMNA (0.65) EPHX2LMNAHDAC4HDAC1HDAC7
SCHEMBL7616443 0.75 LMNA (0.65) EPHX2LMNAHDAC4HDAC1HDAC7
SCHEMBL3461067 0.75 EPHX2 (0.66) EPHX2LMNAHDAC4HDAC1HDAC7
SCHEMBL6361222 0.74 TSHR (0.68) LMNATSHRHPGDSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed