SCHEMBL23979785

SCHEMBL23979785

CN1CCO[C@@H](COC(I)I)C1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.43
PDK1 Q15118 5/20 0.36
IRAK4 Q9NWZ3 1/20 0.34
SLC6A2 P23975 1/20 0.34
EPHA2 P29317 7/20 0.32
KDR P35968 5/20 0.32
EPHB4 P54760 5/20 0.32
EGFR P00533 1/20 0.32
ERBB2 P04626 2/20 0.32
DRD4 P21917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18084612 0.84 HRH3 (0.44) HRH3PDK1IRAK4SLC6A2EPHA2
SCHEMBL24731127 0.84 HRH3 (0.44) HRH3PDK1IRAK4SLC6A2EPHA2
SCHEMBL24730381 0.84 HRH3 (0.44) HRH3PDK1IRAK4SLC6A2EPHA2
SCHEMBL15732028 0.80 HRH3 (0.46) HRH3PDK1IRAK4SLC6A2EPHA2
SCHEMBL3436781 0.78 PDK1 (0.56) HRH3PDK1SLC6A2EPHA2KDR
SCHEMBL7925158 0.78 PDK1 (0.56) HRH3PDK1SLC6A2EPHA2KDR
SCHEMBL12210937 0.78 PDK1 (0.56) HRH3PDK1SLC6A2EPHA2KDR
SCHEMBL25670128 0.77 HRH3 (0.46) HRH3PDK1IRAK4SLC6A2EPHA2
SCHEMBL18773644 0.77 HRH3 (0.46) HRH3PDK1IRAK4SLC6A2EPHA2
SCHEMBL25670134 0.77 HRH3 (0.46) HRH3PDK1IRAK4SLC6A2EPHA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021219072-A1 PREPARATION AND APPLICATION METHOD OF HETEROCYCLIC COMPOUND AS KRAS INHIBITOR 上海科州药物研发有限公司 (CN) 2021-11-04 WO disclosed