SCHEMBL23992191

SCHEMBL23992191

Cc1ccc(C(=O)Nc2ccc(C(F)(F)F)cc2N)nc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 10/20 0.52
KMT2A Q03164 2/20 0.46
BACE1 P56817 2/20 0.46
MEN1 O00255 1/20 0.46
PTGS1 P23219 2/20 0.45
HDAC1 Q13547 8/20 0.45
HDAC2 Q92769 8/20 0.45
NCOR2 Q9Y618 6/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
CFTR P13569 1/20 0.43
BACE2 Q9Y5Z0 1/20 0.42
NCOR1 O75376 1/20 0.42
TRPV1 Q8NER1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23992177 0.83 HDAC1 (0.62) HDAC3HDAC1HDAC2NCOR2NCOR1
SCHEMBL30416650 0.80 HDAC3 (0.63) HDAC3KMT2AMEN1PTGS1HDAC1
SCHEMBL866564 0.80 P2RX1 (0.49) KMT2AMEN1PTGS1HDAC2KDM4E
SCHEMBL27114491 0.77 HDAC1 (0.63) HDAC3KMT2AMEN1HDAC1HDAC2
SCHEMBL1233684 0.77 KCNQ3 (0.60) KMT2ABACE1MEN1PTGS1HDAC1
SCHEMBL16060789 0.76 KDM4E (0.57) KMT2AMEN1PTGS1HDAC1HDAC2
SCHEMBL24086686 0.76 HDAC3 (0.77) HDAC3HDAC1HDAC2NCOR2
SCHEMBL2235637 0.75 CYP1A2 (0.55) HDAC3KMT2AMEN1PTGS1HDAC1
SCHEMBL14967989 0.75 PTGS1 (0.51) HDAC3KMT2APTGS1HDAC1HDAC2
SCHEMBL14453684 0.75 PTGS1 (0.61) HDAC3PTGS1HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021219040-A1 HISTONE DEACETYLASE INHIBITORS FOR IMMUNOMODULATION IN TUMOR MICROENVIRONMENT GNT BIOTECH & MEDICALS CORPORATION (CN) 2021-11-04 WO disclosed