SCHEMBL23993597

SCHEMBL23993597

CC(C)[C@H]1C[C@@H]1c1ccc(C#N)nc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 7/20 0.38
CHRNA7 P36544 2/20 0.35
CHRNB2 P17787 2/20 0.34
CHRNA4 P43681 2/20 0.34
MAOA P21397 1/20 0.34
PIK3CD O00329 1/20 0.32
ABL1 P00519 1/20 0.32
EGFR P00533 1/20 0.32
HCK P08631 1/20 0.32
SRC P12931 1/20 0.32
KDR P35968 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
MTOR P42345 1/20 0.32
EPHB4 P54760 1/20 0.32
PRKDC P78527 1/20 0.32
PI4KB Q9UBF8 1/20 0.32
FASN P49327 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25897312 0.78 KDM1A (0.37) KDM1ACHRNA7CHRNB2CHRNA4CHRNB4
SCHEMBL24867535 0.77 KDM1A (0.40) KDM1ACHRNB2CHRNA4MAOA
SCHEMBL25005549 0.74 GRIA4 (0.46) KDM1AMAOAHRH3
SCHEMBL25005545 0.73 HRH3 (0.43) KDM1ACHRNA7CHRNB2CHRNA4MAOA
SCHEMBL12030737 0.72 DRD2 (0.39) PIK3CDABL1EGFRHCKSRC
SCHEMBL2860558 0.72 KDM4E (0.39) KDM1AFASNELANE
SCHEMBL25004715 0.71 CHRNA7 (0.46) CHRNA7CHRNB2CHRNA4
SCHEMBL30181920 0.70 KDM1A (0.33) KDM1ACHRNA7MAOA
SCHEMBL13596307 0.70 CHRNB2 (0.65) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL3555307 0.69 CHEK1 (0.33) KDM1AFASNELANEADRB1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222522-A1 CD73 INHIBITING 2,4-DIOXOPYRIMIDINE COMPOUNDS GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed