SCHEMBL23993603

SCHEMBL23993603

C[C@H]1C[C@@H]1c1cccc(OC(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
TAS1R2 Q8TE23 1/20 0.44
FFAR1 O14842 1/20 0.43
HTR2A P28223 2/20 0.42
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
KDM1A O60341 1/20 0.40
HCRTR1 O43613 2/20 0.39
HCRTR2 O43614 2/20 0.39
SLC9A1 P19634 1/20 0.39
ADCYAP1R1 P41586 1/20 0.39
EPHX2 P34913 1/20 0.39
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NAMPT P43490 1/20 0.38
NOTUM Q6P988 1/20 0.38
CETP P11597 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12876072 1.00 TAS1R3 (0.44) TAS1R3TAS1R1TAS1R2FFAR1HTR2A
SCHEMBL25004988 0.81 ALOX5 (0.45) TAS1R3TAS1R1TAS1R2FFAR1HTR2A
SCHEMBL23858281 0.80 SSTR1 (0.47) TAS1R3TAS1R1TAS1R2FFAR1HTR2C
SCHEMBL23858279 0.80 SSTR1 (0.47) TAS1R3TAS1R1TAS1R2FFAR1HTR2C
SCHEMBL23858278 0.80 SSTR1 (0.47) TAS1R3TAS1R1TAS1R2FFAR1HTR2C
SCHEMBL30075780 0.80 SSTR1 (0.47) TAS1R3TAS1R1TAS1R2FFAR1HTR2C
SCHEMBL12875677 0.79 KDM1A (0.47) KDM1AEPHX2CYP2D6CYP2C19
SCHEMBL18998726 0.79 KDM1A (0.47) KDM1AEPHX2CYP2D6CYP2C19
SCHEMBL18998470 0.79 KDM1A (0.47) KDM1AEPHX2CYP2D6CYP2C19
SCHEMBL8333649 0.79 HTR2C (0.63) HTR2AHTR2CHTR2BKDM1ASLC9A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222522-A1 CD73 INHIBITING 2,4-DIOXOPYRIMIDINE COMPOUNDS GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed