SCHEMBL24008587

SCHEMBL24008587

FC(F)(F)c1ccc(N2CCCCC2)cn1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.57
MAPT P10636 1/20 0.53
CYP3A4 P08684 3/20 0.50
MAPK1 P28482 2/20 0.49
LMNA P02545 1/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HRH3 Q9Y5N1 1/20 0.48
TRPV4 Q9HBA0 1/20 0.46
PARP1 P09874 1/20 0.43
CHRNB2 P17787 2/20 0.42
CHRNA4 P43681 2/20 0.42
PPARD Q03181 1/20 0.42
PPARA Q07869 1/20 0.42
LCAT P04180 2/20 0.41
CHRM4 P08173 1/20 0.41
NAMPT P43490 1/20 0.40
HSD17B10 Q99714 1/20 0.40
SLC6A9 P48067 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1270114 0.98 DHFR (0.58) DHFRMAPTCYP3A4MAPK1LMNA
SCHEMBL30582922 0.89 DHFR (0.51) DHFRMAPTCYP3A4MAPK1LMNA
SCHEMBL30582912 0.89 DHFR (0.51) DHFRMAPTCYP3A4MAPK1LMNA
SCHEMBL30582875 0.87 DHFR (0.52) DHFRMAPTCYP3A4MAPK1LMNA
SCHEMBL30582888 0.87 DHFR (0.52) DHFRMAPTCYP3A4MAPK1LMNA
SCHEMBL382350 0.83 CHRNB2 (0.58) DHFRMAPTCYP3A4LMNACHRNB2
SCHEMBL31774414 0.83 CHRNB2 (0.58) DHFRMAPTCYP3A4LMNACHRNB2
SCHEMBL13447351 0.83 DHFR (0.58) DHFRMAPTCYP3A4SMN1; SMN2HRH3
SCHEMBL16256660 0.82 MAPT (0.53) DHFRMAPTMAPK1LMNAHTT
Hydrochloric Acid SCHEMBL382186 0.81 CHRNB2 (0.57) DHFRMAPTCYP3A4LMNACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021224864-A1 NON-LYSOSOMAL GLUCOSYLCERAMIDASE INHIBITORS AND USES THEREOF ALECTOS THERAPEUTICS INC. (CA) 2021-11-11 WO disclosed
CN-107001319-B For inhibiting microsomal prostaglandin E2Carboxylic acid compounds of synthase-1 伊莱利利公司 2019-10-01 CN disclosed
CN-107001319-A For inhibiting microsomal prostaglandin E2Carboxylic acid compounds of synthase-1 伊莱利利公司 2017-08-01 CN disclosed