SCHEMBL24009013

SCHEMBL24009013

COc1cncc2c(C)ccnc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.48
CCR5 P51681 2/20 0.48
CCR8 P51685 2/20 0.48
HTR1A P08908 2/20 0.41
ADRA1D P25100 2/20 0.41
ADRA1A P35348 2/20 0.41
ADRA1B P35368 2/20 0.41
PSMD14 O00487 1/20 0.40
COPS5 Q92905 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
CYP17A1 P05093 1/20 0.39
CYP1A2 P05177 1/20 0.39
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
MAOA P21397 2/20 0.37
PDE2A O00408 2/20 0.36
PDE10A Q9Y233 2/20 0.36
PDE4A P27815 2/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18179845 0.79 CCR1 (0.58) CCR1CCR5CCR8HTR1AADRA1D
SCHEMBL24837289 0.78 HTR1A (0.38) HTR1AADRA1DADRA1AADRA1BMAOA
SCHEMBL1337689 0.76 HTR1A (0.61) CCR1CCR5CCR8HTR1AADRA1D
SCHEMBL10257047 0.75 CCR1 (0.48) CCR1CCR5CCR8HTR1AADRA1D
SCHEMBL8032037 0.74 CCR1 (0.69) CCR1CCR5CCR8HTR1AADRA1D
SCHEMBL21064345 0.74 CCR1 (0.52) CCR1CCR5CCR8HTR1AADRA1D
SCHEMBL10290496 0.74 NSD2 (0.50) CCR1CCR5CCR8HTR1AADRA1D
SCHEMBL24009011 0.71 CCR1 (0.46) CCR1CCR5CCR8HTR1AADRA1D
SCHEMBL19660435 0.70 CYP2A6 (0.44) CYP1A2PDE10ACYP19A1ATP4AATP4B
SCHEMBL24838540 0.70 CCR1 (0.57) CCR1CCR5CCR8HTR1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021225969-A1 IMINO SULFANONE INHIBITORS OF ENPP1 VOLASTRA THERAPEUTICS, INC. (US) 2021-11-11 WO disclosed