SCHEMBL24012964

SCHEMBL24012964

Ic1nn(C2CCCCO2)c2ccc(OCCCN(Cc3ccccc3)Cc3ccccc3)cc12

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
KCNA5 P22460 5/20 0.40
MAOB P27338 8/20 0.39
MAOA P21397 6/20 0.39
ACHE P22303 4/20 0.39
BCHE P06276 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30242615 1.00 CYP4F2 (0.41) CYP4F2CYP4A11KCNA5MAOBMAOA
SCHEMBL30242527 0.92 PLA2G2A (0.38) CYP4F2CYP4A11KCNA5MAOBMAOA
SCHEMBL26630592 0.91 CYP4F2 (0.39) CYP4F2CYP4A11KCNA5ACHEBCHE
SCHEMBL24012965 0.90 MAOB (0.41) CYP4F2CYP4A11KCNA5MAOBMAOA
SCHEMBL24012869 0.85 CYP4F2 (0.37) CYP4F2CYP4A11
SCHEMBL24013113 0.85 CYP4F2 (0.52) CYP4F2CYP4A11MAOBMAOA
SCHEMBL24012601 0.85 CYP4F2 (0.37) CYP4F2CYP4A11
SCHEMBL27032051 0.84 CYP4F2 (0.42) CYP4F2CYP4A11MAOBMAOAACHE
SCHEMBL24012649 0.82 CYP4F2 (0.40) CYP4F2CYP4A11
SCHEMBL27032476 0.82 CYP4F2 (0.40) CYP4F2CYP4A11MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357269-A1 NEW MACROCYCLIC LRRK2 KINASE INHIBITORS ONCODESIGN PRECISION MEDICINE (FR) 2023-11-09 US disclosed
US-20230357269-A1 NEW MACROCYCLIC LRRK2 KINASE INHIBITORS ONCODESIGN PRECISION MEDICINE (FR) 2023-11-09 US disclosed
CN-115996932-A New macrocyclic LRRK2 kinase inhibitors 法国施维雅药厂 2023-04-21 CN disclosed
WO-2021224320-A1 NEW MACROCYCLIC LRRK2 KINASE INHIBITORS LES LABORATOIRES SERVIER (FR) 2021-11-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230357269-A1 NEW MACROCYCLIC LRRK2 KINASE INHIBITORS LRRK2, RIN1, GRK3 CYP4F2 4470/4885CYP4A11 4478/4885KCNA5 1961/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.