SCHEMBL24016014

SCHEMBL24016014

CC(=O)NC(c1cccnc1)C1CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.46
NPC1 O15118 1/20 0.46
ALOX12 P18054 1/20 0.46
RAB9A P51151 1/20 0.46
NCOA1 Q15788 1/20 0.46
NCOA3 Q9Y6Q9 1/20 0.46
TSHR P16473 2/20 0.43
HSD17B10 Q99714 2/20 0.43
MAPT P10636 1/20 0.43
KCNA5 P22460 1/20 0.43
CDK2 P24941 1/20 0.41
AKT1 P31749 1/20 0.41
CYP3A4 P08684 3/20 0.41
CYP1A2 P05177 3/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP2C19 P33261 2/20 0.41
OPRM1 P35372 2/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25591483 0.85 NPC1 (0.43) POLBNPC1RAB9ATSHRHSD17B10
SCHEMBL31036989 0.85 NPC1 (0.49) POLBL3MBTL1NPC1ALOX12RAB9A
SCHEMBL30202554 0.81 CYP1A2 (0.57) HSD17B10KCNA5CYP1A2ALDH1A1CYP2C19
SCHEMBL12993111 0.80 MAPT (0.45) TSHRHSD17B10MAPTCYP19A1SMN1; SMN2
SCHEMBL21460469 0.79 ALDH1A1 (0.49) RAB9ATSHRMAPTCDK2AKT1
SCHEMBL20318837 0.79 ALDH1A1 (0.49) RAB9ATSHRMAPTCDK2AKT1
SCHEMBL18228582 0.78 ALDH1A1 (0.46) POLBL3MBTL1TSHRCYP3A4ALDH1A1
SCHEMBL17065013 0.77 CYP3A4 (0.44) POLBL3MBTL1TSHRHSD17B10MAPT
SCHEMBL14392243 0.76 SLC6A4 (0.43) TSHRHSD17B10MAPTCYP3A4CYP1A2
SCHEMBL19322924 0.76 POLB (0.60) POLBKCNA5CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023072974-A1 TRICYCLIC HETEROCYCLES MERCK PATENT GMBH (DE) 2023-05-04 WO disclosed
WO-2021224291-A1 TRICYCLIC HETEROCYCLES USEFUL AS TEAD BINDERS MERCK PATENT GMBH (DE) 2021-11-11 WO disclosed