SCHEMBL24016451

SCHEMBL24016451

O=CN[C@@H](CO)c1ccccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.39
ALDH1A1 P00352 2/20 0.39
KDM4E B2RXH2 2/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
TSHR P16473 2/20 0.38
KCNA5 P22460 2/20 0.37
KCNJ5 P48544 1/20 0.37
KCNJ3 P48549 1/20 0.37
SCN5A Q14524 1/20 0.37
KCND3 Q9UK17 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CYP3A4 P08684 2/20 0.36
TEAD4 Q15561 1/20 0.36
GAA P10253 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP2C19 P33261 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11872592 0.81 EPHX1 (0.53) CYP1A2ALDH1A1KDM4ESLC6A2SLC6A4
SCHEMBL4055323 0.77 TSHR (0.44) CYP1A2ALDH1A1KDM4ESLC6A2SLC6A4
SCHEMBL7126297 0.77 SLC6A2 (0.44) CYP1A2ALDH1A1KDM4ESLC6A2SLC6A4
SCHEMBL27228935 0.77 ALDH1A1 (0.45) CYP1A2ALDH1A1KDM4ESLC6A2SLC6A4
SCHEMBL14630051 0.76 SMN1; SMN2 (0.49) CYP1A2ALDH1A1KDM4ETSHRKCNA5
SCHEMBL24015882 0.75 ALDH1A1 (0.44) CYP1A2ALDH1A1KDM4ESLC6A3TSHR
SCHEMBL19322907 0.75 ALDH1A1 (0.44) CYP1A2ALDH1A1KDM4ESLC6A3TSHR
SCHEMBL24015880 0.75 ALDH1A1 (0.44) CYP1A2ALDH1A1KDM4ESLC6A3TSHR
SCHEMBL12259473 0.75 TSHR (0.42) CYP1A2ALDH1A1KDM4ESLC6A2SLC6A4
SCHEMBL16919267 0.74 CYP1A2 (0.42) CYP1A2ALDH1A1KDM4ESLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023072974-A1 TRICYCLIC HETEROCYCLES MERCK PATENT GMBH (DE) 2023-05-04 WO disclosed
WO-2021224291-A1 TRICYCLIC HETEROCYCLES USEFUL AS TEAD BINDERS MERCK PATENT GMBH (DE) 2021-11-11 WO disclosed