SCHEMBL24030232

SCHEMBL24030232

CCSNc1ccc(Nc2c3ccccc3nc3ccccc23)c(OC)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LY6K Q17RY6 1/20 0.67
KDM1A O60341 7/20 0.64
GLA P06280 2/20 0.64
TOP2B Q02880 2/20 0.64
OPRD1 P41143 2/20 0.64
SLC22A1 O15245 1/20 0.64
ABCC4 O15439 1/20 0.64
NR1I2 O75469 1/20 0.64
TP53 P04637 1/20 0.64
CYP1A2 P05177 1/20 0.64
CYP3A4 P08684 1/20 0.64
CYP2D6 P10635 1/20 0.64
CHRM1 P11229 1/20 0.64
TOP1 P11387 1/20 0.64
TOP2A P11388 1/20 0.64
CYP2C9 P11712 1/20 0.64
DRD2 P14416 1/20 0.64
TSHR P16473 1/20 0.64
ADRA2B P18089 1/20 0.64
ADRA2C P18825 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13524796 0.83 KDM1A (0.72) LY6KKDM1AGLATOP2BOPRD1
SCHEMBL13530937 0.82 KDM1A (0.70) LY6KKDM1AGLATOP2BOPRD1
SCHEMBL24030236 0.81 LY6K (1.00) LY6KKDM1AGLATOP2BOPRD1
SCHEMBL22401407 0.78 LY6K (0.94) LY6KKDM1AGLATOP2BOPRD1
Amsacrine SCHEMBL29360354 0.78 TOP2B (1.00) LY6KKDM1AGLATOP2BOPRD1
Amsacrine SCHEMBL29350869 0.78 TOP2B (1.00) LY6KKDM1AGLATOP2BOPRD1
Amsacrine SCHEMBL28336991 0.78 TOP2B (1.00) LY6KKDM1AGLATOP2BOPRD1
Amsacrine SCHEMBL6256280 0.78 TOP2B (1.00) LY6KKDM1AGLATOP2BOPRD1
Amsacrine SCHEMBL4047 0.78 TOP2B (1.00) LY6KKDM1AGLATOP2BOPRD1
SCHEMBL13529538 0.77 KDM1A (0.67) LY6KKDM1AGLATOP2BOPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021231893-A1 COMPOUNDS FOR INHIBITING LY6K AND METHODS OF USING SAME THE HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE, INC. (US) 2021-11-18 WO disclosed