SCHEMBL24034829

SCHEMBL24034829

CN1C(=O)CCc2cc3c(cc21)OCCC(=O)N3C

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 5/20 0.41
CYP11B2 P19099 7/20 0.39
CYP11B1 P15538 6/20 0.39
CYP19A1 P11511 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP17A1 P05093 1/20 0.39
TRIM24 O15164 3/20 0.37
CYP3A4 P08684 2/20 0.37
KRAS P01116 1/20 0.36
SOS1 Q07889 1/20 0.36
BRD4 O60885 1/20 0.35
CREBBP Q92793 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30076308 0.79 KRAS (0.36) TRPV1CYP11B2CYP11B1KRASSOS1
SCHEMBL23336690 0.78 KRAS (0.37) TRPV1CYP11B2CYP11B1CYP19A1CYP1A2
SCHEMBL24034819 0.77 CD274 (0.37) KRASSOS1
SCHEMBL30076343 0.76 CYP19A1 (0.39) CYP11B2CYP11B1CYP19A1TRIM24CYP3A4
SCHEMBL23336775 0.75 AR (0.38) TRPV1CYP11B2CYP11B1KRASSOS1
SCHEMBL15964517 0.75 KRAS (0.35) CYP11B2CYP11B1KRASSOS1PDE3B
SCHEMBL10274617 0.74 CYP11B2 (0.40) TRPV1CYP11B2CYP11B1KRASSOS1
SCHEMBL23336701 0.74 KRAS (0.34) TRPV1CYP11B2CYP11B1KRASSOS1
SCHEMBL31376465 0.74 POLB (0.39) TRPV1KRASSOS1PDE3BPDE3A
SCHEMBL12713588 0.73 KMO (0.46) PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021228173-A1 AZEPINE FUSED RING COMPOUNDS AND MEDICAL USES THEREOF 中国医药研究开发中心有限公司 2021-11-18 WO disclosed