SCHEMBL2404468

SCHEMBL2404468

O=C(O)c1c(C(F)(F)F)c(-c2ccccc2)nc2ccccc12

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 11/20 0.63
PDE10A Q9Y233 5/20 0.63
LMNA P02545 2/20 0.63
TSHR P16473 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C19 P33261 1/20 0.61
POLB P06746 1/20 0.49
PTGFR P43088 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2404536 0.88 DHODH (0.52) DHODHPDE10ALMNATSHRCYP2D6
Trifluoroacetic Acid SCHEMBL2402411 0.85 DHODH (0.49) DHODHPDE10ALMNATSHRCYP2D6
SCHEMBL29290337 0.80 DHODH (0.69) DHODHPDE10ALMNATSHRCYP2D6
SCHEMBL2429278 0.79 PDE10A (0.45) DHODHPDE10ALMNATSHRCYP2D6
SCHEMBL28048083 0.78 LMNA (0.49) DHODHPDE10ALMNATSHRCYP2C19
SCHEMBL24122754 0.78 LMNA (1.00) DHODHPDE10ALMNATSHRCYP2D6
SCHEMBL3908668 0.78 DHODH (0.71) DHODHPDE10ALMNATSHRCYP2D6
Oxycinchophen SCHEMBL1170683 0.78 DHODH (1.00) DHODHPDE10ALMNATSHRCYP2D6
Oxycinchophen SCHEMBL29460357 0.78 DHODH (1.00) DHODHPDE10ALMNATSHRCYP2D6
Oxycinchophen SCHEMBL31654029 0.78 DHODH (1.00) DHODHPDE10ALMNATSHRCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2549872-A1 TRPV4 ANTAGONISTS GlaxoSmithKline LLC (US) 2013-01-30 EP disclosed
WO-2011119704-A1 TRPV4 ANTAGONISTS GLAXOSMITHKLINE LLC (US) 2011-09-29 WO disclosed
WO-2011119701-A1 TRPV4 ANTAGONISTS GLAXOSMITHKLINE LLC (US) 2011-09-29 WO disclosed