SCHEMBL28048083

SCHEMBL28048083

FC(F)(F)c1c(-c2ccccc2)nc2ccccc2c1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.49
ESR1 P03372 4/20 0.47
ESR2 Q92731 2/20 0.45
TOP1 P11387 1/20 0.44
NUDT1 P36639 2/20 0.44
ADORA2A P29274 2/20 0.43
ENPP1 P22413 1/20 0.42
KDM4E B2RXH2 3/20 0.42
PKM P14618 1/20 0.42
PDE10A Q9Y233 2/20 0.41
DHODH Q02127 1/20 0.41
TSHR P16473 2/20 0.41
HTT P42858 1/20 0.41
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4364503 0.79 TOP1 (0.44) LMNATOP1NUDT1ADORA2AKDM4E
SCHEMBL2404468 0.78 DHODH (0.63) LMNAPDE10ADHODHTSHRPOLB
SCHEMBL971895 0.77 LMNA (0.62) LMNAESR1ESR2NUDT1ADORA2A
SCHEMBL27909470 0.77 LMNA (0.53) LMNAESR1ESR2NUDT1ADORA2A
SCHEMBL27810976 0.76 LMNA (0.61) LMNAESR1ESR2NUDT1ADORA2A
SCHEMBL28239158 0.76 LMNA (0.61) LMNAESR1ESR2NUDT1ADORA2A
SCHEMBL2404536 0.75 DHODH (0.52) LMNAPDE10ADHODHTSHRGAA
SCHEMBL28962062 0.74 NUDT1 (0.58) LMNAESR1ESR2NUDT1ADORA2A
SCHEMBL28048054 0.74 TACR3 (0.48) NUDT1KDM4EPDE10ATSHRGAA
SCHEMBL13758058 0.73 PDE10A (0.60) LMNAESR1ESR2TOP1NUDT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105175327-B A kind of synthetic method of quinoline 南阳师范学院 2017-07-14 CN disclosed
CN-105175327-A Synthesis method of quinoline derivatives UNIV NANYANG NORMAL 2015-12-23 CN disclosed