SCHEMBL24072579

SCHEMBL24072579

Cc1cc(C(C)(C)N2CCN(C)CC2)no1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
HRH4 Q9H3N8 3/20 0.33
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
CSF1R P07333 1/20 0.31
KMT2A Q03164 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23966639 0.83 MEN1 (0.37) HRH4CSF1RKMT2A
SCHEMBL25799458 0.81 SMN1; SMN2 (0.34) ALDH1A1HRH4TSHRKMT2A
SCHEMBL427051 0.69 ALDH1A1 (0.43) ALDH1A1KDM4ETRPM8
SCHEMBL20234660 0.68 ALDH1A1 (0.47) ALDH1A1KDM4EHRH4CYP1A2CYP2C9
SCHEMBL10104245 0.66 TRPM8 (0.38) ALDH1A1KDM4ETSHRMAPK1KMT2A
SCHEMBL20320491 0.66 TRPM8 (0.38) ALDH1A1KDM4ECYP1A2TSHRTRPM8
SCHEMBL1089518 0.66 TRPM8 (0.38) ALDH1A1KDM4ETSHRKMT2ATRPM8
SCHEMBL13559779 0.66 AURKA (0.53) ALDH1A1KDM4E
SCHEMBL19599660 0.64 KDM4E (0.51) ALDH1A1KDM4ECYP1A2
SCHEMBL27360043 0.64 SMN1; SMN2 (0.41) ALDH1A1HRH4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021252488-A1 INHIBITORS OF NEK7 KINASE Halia Therapeutics, Inc. (US) 2021-12-16 WO disclosed
WO-2021242505-A1 INHIBITORS OF NEK7 KINASE Halia Therapeutics, Inc. (US) 2021-12-02 WO disclosed