SCHEMBL2408897

SCHEMBL2408897

CN(C(=O)Cc1ccc(C(F)(F)F)cc1)C1CC1

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 12/20 0.69
GPR119 Q8TDV5 11/20 0.63
CCR5 P51681 4/20 0.62
PTGDR2 Q9Y5Y4 1/20 0.53
OPRK1 P41145 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3527812 0.83 KCNH2 (0.55) KCNH2GPR119CCR5PTGDR2OPRK1
SCHEMBL2404203 0.82 CCR5 (0.65) KCNH2GPR119CCR5OPRK1
Hydrochloric Acid SCHEMBL11528044 0.82 KCNH2 (0.54) KCNH2GPR119CCR5PTGDR2OPRK1
SCHEMBL2407533 0.82 KCNH2 (0.49) KCNH2GPR119CCR5
SCHEMBL2405156 0.82 CCR5 (0.60) KCNH2GPR119CCR5
SCHEMBL18388186 0.82 HDAC4 (0.54) KCNH2GPR119CCR5OPRK1
SCHEMBL13434079 0.80 CCR5 (0.63) KCNH2CCR5PTGDR2
SCHEMBL2405257 0.78 CCR5 (0.62) CCR5PTGDR2
SCHEMBL2406788 0.78 CCR5 (0.62) KCNH2GPR119CCR5
Hydrochloric Acid SCHEMBL5630464 0.77 SIGMAR1 (0.71) OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110212968-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD. (CH) 2011-09-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110212968-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES HCRTR2, HCRTR1, HRH3 KCNH2 498/4885GPR119 60/4885CCR5 2055/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.