SCHEMBL24101477

SCHEMBL24101477

CC1=C(CC(=O)O)c2cc(F)ccc2/C1=C\c1ccc(S(=O)(=O)c2ccc(F)cc2)cc1

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 14/20 0.84
CYP1A2 P05177 3/20 0.83
MAPT P10636 3/20 0.83
MAPK1 P28482 3/20 0.83
TDP1 Q9NUW8 2/20 0.83
CYP3A4 P08684 2/20 0.83
PMP22 Q01453 2/20 0.83
NPSR1 Q6W5P4 2/20 0.83
GLA P06280 1/20 0.83
TSHR P16473 1/20 0.83
EDNRA P25101 1/20 0.83
HIF1A Q16665 1/20 0.83
HSD17B10 Q99714 1/20 0.83
RXRA P19793 6/20 0.74
PTGS2 P35354 2/20 0.71
EGFR P00533 1/20 0.71
ADORA3 P0DMS8 1/20 0.71
DRD1 P21728 1/20 0.71
PTGS1 P23219 1/20 0.71
OPRM1 P35372 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30095195 1.00 PPARG (0.84) PPARGCYP1A2MAPTMAPK1TDP1
SCHEMBL30913371 0.92 CYP1A2 (0.74) PPARGCYP1A2MAPTMAPK1TDP1
Exisulind SCHEMBL4776597 0.91 CYP1A2 (1.00) PPARGCYP1A2MAPTMAPK1TDP1
Exisulind SCHEMBL25371 0.91 CYP1A2 (1.00) PPARGCYP1A2MAPTMAPK1TDP1
Exisulind SCHEMBL29395528 0.91 CYP1A2 (1.00) PPARGCYP1A2MAPTMAPK1TDP1
Exisulind SCHEMBL1651133 0.91 CYP1A2 (1.00) PPARGCYP1A2MAPTMAPK1TDP1
SCHEMBL30913530 0.91 PPARG (0.74) PPARGCYP1A2MAPTMAPK1TDP1
Exisulind SCHEMBL9711060 0.90 CYP1A2 (0.98) PPARGCYP1A2MAPTMAPK1TDP1
SCHEMBL8521006 0.90 CYP1A2 (0.82) PPARGCYP1A2MAPTMAPK1TDP1
Exisulind SCHEMBL7634644 0.90 CYP1A2 (0.98) PPARGCYP1A2MAPTMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230234909-A1 INDENE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR THERAPEUTIC APPLICATIONS NUCMITO PHARMACEUTICALS CO. LTD. (CN) 2023-07-27 US claimed
CN-116472034-A Indene compound, pharmaceutical composition thereof and therapeutic application thereof 藤济(厦门)生物医药科技有限公司 2023-07-21 CN claimed
CN-117916215-A Indene compound, pharmaceutical composition thereof and therapeutic application thereof 藤济(厦门)生物医药科技有限公司 2024-04-19 CN disclosed
US-20240116845-A1 INDENE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR THERAPEUTIC APPLICATIONS NUCMITO PHARMACEUTICALS CO LTD (CN) 2024-04-11 US disclosed
US-20230234909-A1 INDENE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR THERAPEUTIC APPLICATIONS NUCMITO PHARMACEUTICALS CO. LTD. (CN) 2023-07-27 US disclosed
US-20230234909-A1 INDENE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR THERAPEUTIC APPLICATIONS NUCMITO PHARMACEUTICALS CO. LTD. (CN) 2023-07-27 US disclosed
US-20230234909-A1 INDENE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR THERAPEUTIC APPLICATIONS NUCMITO PHARMACEUTICALS CO. LTD. (CN) 2023-07-27 US disclosed
CN-116472034-A Indene compound, pharmaceutical composition thereof and therapeutic application thereof 藤济(厦门)生物医药科技有限公司 2023-07-21 CN disclosed
WO-2021249529-A1 INDENE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR THERAPEUTIC APPLICATIONS NUCMITO PHARMACEUTICALS CO., LTD. (CN) 2021-12-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230234909-A1 INDENE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR THERAPEUTIC APPLICATIONS MMP1, IDO1, COL1A1 PPARG 378/4885CYP1A2 24/4885MAPT 1585/4885
US-20240116845-A1 INDENE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR THERAPEUTIC APPLICATIONS MMP1, IDO1, COL1A1 PPARG 378/4885CYP1A2 24/4885MAPT 1585/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.