SCHEMBL2412263

SCHEMBL2412263

CNC(=O)COC(=O)NCCCCc1cc(-c2ccc(Cl)cc2)nc(C2CC2)n1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.38
POLB P06746 2/20 0.37
PDE4B Q07343 3/20 0.36
PDE4D Q08499 3/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ADORA3 P0DMS8 2/20 0.34
MAPT P10636 4/20 0.34
PSD A5PKW4 1/20 0.34
TP53 P04637 2/20 0.33
CTRC Q99895 1/20 0.33
RECQL P46063 1/20 0.33
VCP P55072 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2416165 0.88 POLB (0.38) POLBKDM4EALDH1A1ADORA3MAPT
SCHEMBL2411224 0.87 POLB (0.40) FAAHPOLBKDM4EALDH1A1ADORA3
SCHEMBL2411128 0.85 POLB (0.38) POLBKDM4EALDH1A1ADORA3MAPT
SCHEMBL2413838 0.84 POLB (0.40) FAAHPOLBKDM4EALDH1A1ADORA3
SCHEMBL2843229 0.83 PDE4B (0.43) PDE4BPDE4DKDM4EMAPTPSD
SCHEMBL2410278 0.83 POLB (0.40) FAAHPOLBKDM4EALDH1A1MAPT
SCHEMBL2409791 0.81 POLB (0.40) POLBKDM4EALDH1A1ADORA3MAPT
SCHEMBL2408187 0.80 POLB (0.40) FAAHPOLBKDM4EALDH1A1ADORA3
SCHEMBL2409167 0.79 POLB (0.42) POLBKDM4EALDH1A1ADORA3MAPT
SCHEMBL2413367 0.79 MAPT (0.53) POLBALDH1A1MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110237595-A1 DERIVATIVES OF HETEROARYL-ALKYLCARBAMATES, METHODS FOR THEIR PREPARATION AND USE THEREOF AS FATTY ACID AMIDO HYDROLASE ENZYME INHIBITORS SANOFI-AVENTIS (FR) 2011-09-29 US disclosed
US-20100069405-A1 DERIVATIVES OF HETEROARYL-ALKYLCARBAMATES, METHODS FOR THEIR PREPARATION AND USE THEREOF AS FATTY ACID AMIDO HYDROLASE ENZYME INHIBITORS SANOFI-AVENTIS (FR) 2010-03-18 US disclosed
US-7645757-B2 Derivatives of heteroaryl-alkylcarbamates, methods for their preparation and use thereof as fatty acid amido hydrolase enzyme inhibitors SANOFI-AVENTIS (FR) 2010-01-12 US disclosed
US-20070021426-A1 DERIVATIVES OF HETEROARYL-ALKYLCARBAMATES, METHODS FOR THEIR PREPARATION AND USE THEREOF AS FATTY ACID AMIDO HYDROLASE ENZYME INHIBITORS SANOFI-AVENTIS (FR) 2007-01-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110237595-A1 DERIVATIVES OF HETEROARYL-ALKYLCARBAMATES, METHODS FOR THEIR PREPARATION AND USE THEREOF AS FATTY ACID AMIDO HYDROLASE ENZYME INHIBITORS FAAH, FAAH2, CNR1 FAAH 1/4885POLB 2741/4885PDE4B 2310/4885
US-20100069405-A1 DERIVATIVES OF HETEROARYL-ALKYLCARBAMATES, METHODS FOR THEIR PREPARATION AND USE THEREOF AS FATTY ACID AMIDO HYDROLASE ENZYME INHIBITORS FAAH, FAAH2, CNR1 FAAH 1/4885POLB 2741/4885PDE4B 2310/4885
US-20070021426-A1 DERIVATIVES OF HETEROARYL-ALKYLCARBAMATES, METHODS FOR THEIR PREPARATION AND USE THEREOF AS FATTY ACID AMIDO HYDROLASE ENZYME INHIBITORS FAAH, FAAH2, CNR2 FAAH 1/4885POLB 1835/4885PDE4B 2908/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.