SCHEMBL24123750

SCHEMBL24123750

COc1cc(C)cc(N2CCN(C)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.51
FFAR4 Q5NUL3 1/20 0.47
HTR3A P46098 1/20 0.46
DNMT1 P26358 1/20 0.45
RAD52 P43351 1/20 0.45
PHGDH O43175 1/20 0.45
DRD2 P14416 3/20 0.44
HTR1A P08908 1/20 0.44
HTR2A P28223 1/20 0.44
HTR7 P34969 1/20 0.44
ADRA1A P35348 1/20 0.44
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
ADRA2C P18825 2/20 0.43
SIRT6 Q8N6T7 1/20 0.43
KDM4E B2RXH2 2/20 0.43
TGFBR1 P36897 1/20 0.43
ACVR1 Q04771 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23657292 0.89 ADRB1 (0.58) ADRB1HTR3ADRD2NPC1RAB9A
SCHEMBL13928098 0.85 ADRB1 (0.55) ADRB1FFAR4HTR3APHGDHNPC1
SCHEMBL12359403 0.82 MAPT (0.54) HTR3AHTR1ANPC1RAB9AADRA2C
SCHEMBL17144207 0.82 ADRB1 (0.56) ADRB1HTR3AKDM4EALDH1A1GFER
SCHEMBL23657169 0.81 ADRB1 (0.50) ADRB1FFAR4HTR3ADRD2NPC1
SCHEMBL23657300 0.81 ADRB1 (0.50) ADRB1HTR3ADRD2NPC1RAB9A
SCHEMBL10127523 0.81 ADRA2C (0.59) ADRB1HTR3ARAD52NPC1RAB9A
SCHEMBL2873315 0.81 ADRB1 (0.80) ADRB1HTR3AHTR1ATGFBR1ACVR1
SCHEMBL14032316 0.81 PRKDC (0.52) ADRB1FFAR4NPC1RAB9AKDM4E
SCHEMBL10104342 0.80 FFAR4 (0.51) FFAR4HTR3APHGDHNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4169919-A1 PYRAZOLO[3,4-D]PYRIMIDINE-3-KETONE DERIVATIVE AS WEE-1 INHIBITOR Wigen Biomedicine Technology (Shanghai) Co., Ltd. (CN) 2023-04-26 EP disclosed
WO-2021254389-A1 PYRAZOLO[3,4-D]PYRIMIDINE-3-KETONE DERIVATIVE AS WEE-1 INHIBITOR 微境生物医药科技(上海)有限公司 2021-12-23 WO disclosed