SCHEMBL2412641

SCHEMBL2412641

CN(Cc1cc(-c2cccnc2C#N)n(S(=O)(=O)c2ccccc2)c1)C(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 4/20 0.37
SLC6A4 P31645 4/20 0.37
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
GLS O94925 1/20 0.33
F2 P00734 2/20 0.33
HTR6 P50406 2/20 0.33
PLCG1 P19174 1/20 0.32
TNF P01375 3/20 0.32
RORC P51449 1/20 0.32
PDK2 Q15119 1/20 0.31
KMT2A Q03164 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4427592 0.95 HTR2C (0.34) HTR2CSLC6A4CTSLCTSBCTSS
SCHEMBL2410003 0.90 HTR2C (0.34) HTR2CSLC6A4CTSLCTSBCTSS
SCHEMBL2414628 0.90 TACR1 (0.35) HTR2CSLC6A4CTSLCTSBCTSS
SCHEMBL2406675 0.90 HTR2C (0.34) HTR2CSLC6A4CTSLCTSBCTSS
SCHEMBL2417461 0.90 GLS (0.32) HTR2CSLC6A4GLSPLCG1
SCHEMBL2411191 0.90 HTR2C (0.31) HTR2CSLC6A4PLCG1
SCHEMBL2409829 0.90 HTR2C (0.35) HTR2CSLC6A4CTSLCTSBCTSS
SCHEMBL2408479 0.89 HTR6 (0.36) HTR6TNFKMT2APTGDR2LMNA
SCHEMBL2410418 0.88 RET (0.33) HTR2CSLC6A4PLCG1RORCPTGDR2
SCHEMBL2415723 0.88 HTR2C (0.39) HTR2CSLC6A4GLSF2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed