SCHEMBL24129192

SCHEMBL24129192

Cc1nc2ncnn2c(C2CC2)c1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.46
PAX2 Q02962 1/20 0.43
ALDH1A1 P00352 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
HSD17B10 Q99714 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
MAPK1 P28482 2/20 0.42
USP2 O75604 2/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
ALOX15 P16050 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.39
MAPT P10636 3/20 0.39
HTT P42858 2/20 0.39
KDM4E B2RXH2 3/20 0.39
HPGD P15428 1/20 0.39
ENPP1 P22413 2/20 0.38
NPC1 O15118 1/20 0.38
GALR3 O60755 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL353089 0.74 HSD17B10 (0.55) TSHRPAX2ALDH1A1MEN1KMT2A
SCHEMBL24129332 0.74 PAX2 (0.50) TSHRPAX2ALDH1A1MEN1KMT2A
SCHEMBL31557748 0.73 TSHR (0.56) TSHRPAX2ALDH1A1MEN1KMT2A
SCHEMBL976541 0.72 MAPK1 (0.39) TSHRALDH1A1KMT2AMAPK1LMNA
SCHEMBL14271003 0.72 KDM4E (0.48) TSHRPAX2ALDH1A1HSD17B10KDM4E
SCHEMBL24129389 0.72 ENPP1 (0.46) TSHRPAX2ALDH1A1MEN1KMT2A
SCHEMBL10407276 0.72 TSHR (0.50) TSHRPAX2ALDH1A1MEN1KMT2A
SCHEMBL22968432 0.72 TSHR (0.50) TSHRPAX2ALDH1A1ENPP1
SCHEMBL10407277 0.72 TSHR (0.50) TSHRPAX2ALDH1A1MEN1KMT2A
SCHEMBL5199168 0.72 TSHR (0.50) TSHRPAX2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021257614-A1 HETEROCYCLIC INHIBITORS OF ENPP1 VOLASTRA THERAPEUTICS, INC. (US) 2021-12-23 WO disclosed