SCHEMBL2413477

SCHEMBL2413477

CC1C(C(=O)O)CN1Cc1cccc(-c2cc3cc(Cc4ccccc4)ccc3o2)c1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 9/20 0.59
S1PR3 Q99500 4/20 0.55
KCNH2 Q12809 1/20 0.53
MAOB P27338 8/20 0.49
MAOA P21397 2/20 0.49
FFAR1 O14842 2/20 0.44
CYP26A1 O43174 1/20 0.44
CYP26B1 Q9NR63 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1602296 0.82 S1PR1 (0.85) S1PR1S1PR3KCNH2
SCHEMBL12319320 0.81 S1PR1 (0.63) S1PR1S1PR3KCNH2MAOBMAOA
SCHEMBL1601740 0.79 S1PR1 (0.68) S1PR1S1PR3KCNH2MAOBMAOA
SCHEMBL1601626 0.78 S1PR1 (0.61) S1PR1S1PR3KCNH2MAOB
SCHEMBL12318147 0.77 S1PR1 (0.63) S1PR1S1PR3KCNH2MAOBMAOA
SCHEMBL2414430 0.74 S1PR1 (0.67) S1PR1S1PR3KCNH2
SCHEMBL1603237 0.74 S1PR1 (1.00) S1PR1S1PR3KCNH2
SCHEMBL9543098 0.73 MAPT (0.50) S1PR1
SCHEMBL2420094 0.73 S1PR1 (0.54) S1PR1S1PR3KCNH2MAOBMAOA
SCHEMBL2415217 0.72 S1PR1 (0.53) S1PR1S1PR3KCNH2MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364976-A1 S1P receptor modulating compounds and use thereof EPIX Pharmaceuticals, Inc. (US) 2011-09-14 EP disclosed