SCHEMBL24159059

SCHEMBL24159059

CNC(=O)CCCC(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.43
ALDH1A1 P00352 1/20 0.36
RECQL P46063 1/20 0.34
PDK2 Q15119 2/20 0.34
CNR1 P21554 2/20 0.33
CNR2 P34972 2/20 0.33
MCL1 Q07820 1/20 0.33
POLB P06746 1/20 0.33
MPO P05164 1/20 0.33
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32
FAAH O00519 1/20 0.31
HSP90AA1 P07900 1/20 0.31
OXER1 Q8TDS5 1/20 0.31
MTNR1A P48039 1/20 0.31
NAMPT P43490 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9363475 0.88 LMNA (0.48) LMNAALDH1A1PDK2CNR1CNR2
SCHEMBL12745317 0.79 LMNA (0.44) LMNAALDH1A1RECQLCNR1CNR2
SCHEMBL18555743 0.77 KDM4E (0.44) LMNAALDH1A1POLBHDAC3HDAC1
SCHEMBL7753090 0.77 LMNA (0.57) LMNAALDH1A1RECQLMCL1POLB
SCHEMBL5909180 0.77 LMNA (0.57) LMNARECQLMCL1POLBHDAC3
SCHEMBL21078328 0.76 LMNA (0.46) LMNAALDH1A1PDK2CNR1CNR2
Hydrochloric Acid SCHEMBL375176 0.76 KDM4E (0.43) LMNAALDH1A1POLBHDAC3HDAC1
SCHEMBL14963638 0.75 LMNA (0.50) LMNAALDH1A1RECQLPDK2CNR1
SCHEMBL5909483 0.75 HDAC3 (0.55) LMNARECQLMCL1HDAC3HDAC1
SCHEMBL5909431 0.75 HDAC3 (0.55) LMNARECQLMCL1HDAC3HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3793565-B1 MCL-1 INHIBITORS GILEAD SCIENCES INC (US) 2022-01-05 EP disclosed