SCHEMBL24178458

SCHEMBL24178458

C[C@@H](N)CC#C[Si](C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.39
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23153952 1.00 HTR2A (0.39) HTR2AALDH1A1
SCHEMBL10094588 0.78
SCHEMBL15755391 0.74 TSHR (0.32) ALDH1A1
SCHEMBL15755393 0.74 TSHR (0.32) ALDH1A1
SCHEMBL7928919 0.69
SCHEMBL26996497 0.69
SCHEMBL21846946 0.69 HTR2A (0.43) HTR2AALDH1A1
SCHEMBL4544179 0.69
SCHEMBL28027671 0.68
SCHEMBL24178278 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12448386-B2 Processes for the preparation of substituted 1,3,4,9-tetrahydro-2H-pyrido[3,4-b]indoles HOFFMANN-LA ROCHE INC. (US) 2025-10-21 US disclosed
US-11873305-B2 Processes for synthesis of substituted indole intermediates for the synthesis of serd compounds GENENTECH, INC. (US) 2024-01-16 US disclosed
US-11873305-B2 Processes for synthesis of substituted indole intermediates for the synthesis of serd compounds GENENTECH, INC. (US) 2024-01-16 US disclosed
CN-115916750-A Process for preparing SERD tricyclic compounds having substituted phenyl or pyridyl moieties 基因泰克公司 2023-04-04 CN disclosed
US-20220002304-A1 PROCESSES FOR MAKING SERD TRICYCLIC COMPOUNDS HAVING A SUBSTITUTED PHENYL OR PYRIDINYL MOIETY GENENTECH, INC. (US) 2022-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11873305-B2 Processes for synthesis of substituted indole intermediates for the synthesis of serd compounds WEE1, WEE2, INMT HTR2A 728/4885ALDH1A1 2335/4885
US-20220002304-A1 PROCESSES FOR MAKING SERD TRICYCLIC COMPOUNDS HAVING A SUBSTITUTED PHENYL OR PYRIDINYL MOIETY PLK2, CHEK1, PLK4 HTR2A 986/4885ALDH1A1 1315/4885
US-12448386-B2 Processes for the preparation of substituted 1,3,4,9-tetrahydro-2H-pyrido[3,4-b]indoles WEE1, WEE2, PGK1 HTR2A 337/4885ALDH1A1 3168/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.