SCHEMBL24182136

SCHEMBL24182136

CCn1cc(C(C)O)c2cc(Cl)ccc21

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.56
CYP19A1 P11511 4/20 0.47
CYP2C19 P33261 2/20 0.44
PTGER4 P35408 1/20 0.38
KDM1A O60341 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
RAD52 P43351 1/20 0.36
NLRP1 Q9C000 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27418241 0.78 CYP19A1 (0.43) KCNH2CYP19A1CYP2C19PTGER4MAPT
SCHEMBL24824867 0.77 PTGER4 (0.44) KCNH2CYP19A1CYP2C19PTGER4PTGDR2
SCHEMBL27693251 0.76 PSEN1 (0.41) KCNH2CYP19A1CYP2C19KDM1A
SCHEMBL10467514 0.76 PSEN1 (0.41) KCNH2CYP19A1CYP2C19KDM1A
SCHEMBL16727205 0.76 PTGER4 (0.43) KCNH2CYP19A1CYP2C19PTGER4PTGDR2
SCHEMBL27693102 0.74 CYP19A1 (0.41) CYP19A1CYP2C19PTGDR2
SCHEMBL18015838 0.74 KCNH2 (0.56) KCNH2CYP19A1CYP2C19PTGER4PTGDR2
SCHEMBL13153267 0.74 PTGER4 (0.42) KCNH2CYP19A1CYP2C19PTGER4PTGDR2
SCHEMBL12485507 0.73 KDM4E (0.54) KCNH2PTGDR2CYP1A2TDP1
SCHEMBL22450724 0.73 KCNH2 (0.56) KCNH2PTGER4PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3936126-A1 COMBINATION OF IAP INHIBITOR AND IMMUNE CHECKPOINT INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2022-01-12 EP disclosed