SCHEMBL27693102

SCHEMBL27693102

CCn1cc(C(C)C(N=C=O)C(=O)O)c2cc(Cl)ccc21

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.41
KDM4E B2RXH2 1/20 0.36
PSEN1 P49768 3/20 0.36
PSEN2 P49810 2/20 0.36
APH1B Q8WW43 2/20 0.36
NCSTN Q92542 2/20 0.36
APH1A Q96BI3 2/20 0.36
PSENEN Q9NZ42 2/20 0.36
CYP2C19 P33261 1/20 0.36
CPT1A P50416 2/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
HAT1 O14929 2/20 0.35
EP300 Q09472 2/20 0.35
CPT2 P23786 1/20 0.35
CPT1B Q92523 1/20 0.35
CNR1 P21554 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27674773 0.87 LMNA (0.43) CYP19A1KDM4ECYP2C19
SCHEMBL24182136 0.74 KCNH2 (0.56) CYP19A1CYP2C19PTGDR2
SCHEMBL27693251 0.73 PSEN1 (0.41) CYP19A1KDM4EPSEN1PSEN2APH1B
SCHEMBL10467514 0.73 PSEN1 (0.41) CYP19A1KDM4EPSEN1PSEN2APH1B
SCHEMBL10773483 0.72 TRPA1 (0.40) CYP19A1KDM4ECPT1ACPT2CPT1B
SCHEMBL10468207 0.72 TRPA1 (0.40) CYP19A1KDM4ECPT1ACPT2CPT1B
SCHEMBL10773430 0.72 CYP19A1 (0.35) CYP19A1KDM4EPSEN1PSEN2APH1B
SCHEMBL12485507 0.69 KDM4E (0.54) KDM4EPTGDR2HAT1EP300CNR1
SCHEMBL27418241 0.69 CYP19A1 (0.43) CYP19A1KDM4EPSEN1PSEN2APH1B
SCHEMBL10773477 0.68 CYP19A1 (0.36) CYP19A1KDM4EPSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-87103087-A As diethylenediamine compound of platelet activation factor-antagonist and preparation method thereof 1987-11-04 CN disclosed