SCHEMBL24192519

SCHEMBL24192519

CN(CCOCCn1nccc1B1OC(C)(C)C(C)(C)O1)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 1/20 0.36
PDK2 Q15119 1/20 0.34
BACE1 P56817 1/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
AAK1 Q2M2I8 3/20 0.31
KAT6A Q92794 1/20 0.31
KAT5 Q92993 1/20 0.31
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31
HTR2C P28335 1/20 0.31
SLC6A4 P31645 1/20 0.31
FPR3 P25089 1/20 0.30
FPR2 P25090 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25969633 0.91 USP30 (0.37) USP30BACE1BACE2AAK1PRMT5
SCHEMBL25969661 0.87 USP30 (0.37) USP30PDK2BACE1BACE2AAK1
SCHEMBL25969622 0.81 USP30 (0.39) USP30BACE1BACE2AAK1PRMT5
SCHEMBL25969654 0.80 USP30 (0.37) USP30BACE1BACE2AAK1PRMT5
SCHEMBL25345280 0.78 PDK2 (0.34) PDK2AAK1KAT6AKAT5HTR2C
SCHEMBL26924166 0.76 USP30 (0.39) USP30PDK2AAK1
SCHEMBL25341995 0.74 USP30 (0.34) USP30PDK2
SCHEMBL30568630 0.74 USP30 (0.34) USP30PDK2
SCHEMBL26924205 0.73 USP30 (0.41) USP30PDK2BACE1BACE2AAK1
SCHEMBL25969641 0.73 USP30 (0.39) USP30BACE1BACE2AAK1PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230257396-A1 MACROCYCLES AND THEIR USE BLOSSOMHILL THERAPEUTICS INC (US) 2023-08-17 US disclosed
US-20230257396-A1 MACROCYCLES AND THEIR USE BLOSSOMHILL THERAPEUTICS INC (US) 2023-08-17 US disclosed
WO-2022011123-A1 MACROCYCLES AND THEIR USE BLOSSOMHILL THERAPEUTICS, INC. (US) 2022-01-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230257396-A1 MACROCYCLES AND THEIR USE VHL, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, DLD USP30 4382/4885PDK2 580/4885BACE1 2544/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.