SCHEMBL24201621

SCHEMBL24201621

COc1cc(C)c2c(c1CN1CCCCC1)CCN2

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.47
GAA P10253 1/20 0.42
ALDH1A1 P00352 2/20 0.41
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41
KDM4E B2RXH2 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.38
CFB P00751 1/20 0.38
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24054518 0.83 ACHE (0.38) PARP1
SCHEMBL25648517 0.83 CFB (0.39) PARP1CFB
SCHEMBL25648972 0.79 PARP1 (0.44) PARP1CFB
SCHEMBL23783633 0.73 GAA (0.54) GAAALDH1A1MEN1TSHRKMT2A
SCHEMBL6314736 0.73 HTR2A (0.36) PARP1GAAALDH1A1KDM4ETDP1
SCHEMBL23863696 0.71 CFB (0.48) GAAALDH1A1MEN1TSHRKMT2A
SCHEMBL23641611 0.70 HTR2A (0.37) PARP1GAAALDH1A1KDM4EPOLB
SCHEMBL1427544 0.70 GAA (0.55) GAAALDH1A1MEN1TSHRKMT2A
SCHEMBL19446025 0.69 CFB (0.74) CFB
SCHEMBL24201510 0.68 MEN1 (0.46) GAAALDH1A1MEN1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3939591-A1 QUINAZOLINE AND INDOLE COMPOUNDS TO TREAT MEDICAL DISORDERS Achillion Pharmaceuticals, Inc. (US) 2022-01-19 EP disclosed