SCHEMBL24201665

SCHEMBL24201665

CCCCNC(=O)/C(C)=N/c1c(C)ncnc1N1CCc2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 11/20 0.47
MKNK2 Q9HBH9 11/20 0.47
EIF4E P06730 1/20 0.45
LMNA P02545 2/20 0.42
HTT P42858 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
TP53 P04637 1/20 0.40
THRB P10828 1/20 0.40
EGFR P00533 2/20 0.39
ACKR3 P25106 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23761494 0.92 MKNK1 (0.44) MKNK1MKNK2EIF4EHTTEGFR
SCHEMBL24201911 0.88 MKNK1 (0.42) MKNK1MKNK2EIF4ELMNAHTT
SCHEMBL24201968 0.88 MKNK1 (0.42) MKNK1MKNK2EIF4ELMNAHTT
SCHEMBL23761516 0.84 MKNK1 (0.40) MKNK1MKNK2EIF4EHTTEGFR
SCHEMBL24201884 0.82 MKNK1 (0.39) MKNK1MKNK2EIF4EHTTALDH1A1
SCHEMBL23761514 0.81 ALDH1A1 (0.41) LMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL23761323 0.80 MKNK1 (0.48) MKNK1MKNK2EIF4ELMNA
SCHEMBL23761540 0.79 MKNK1 (0.36) MKNK1MKNK2EIF4ELMNAHTT
SCHEMBL23761404 0.78 MKNK1 (0.43) MKNK1MKNK2EIF4EHTTMAPT
SCHEMBL24201824 0.78 MKNK1 (0.45) MKNK1MKNK2EIF4ELMNAEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3939981-A1 FUSED THIAZOLOPYRIMIDINE DERIVATIVES AS MNKS INHIBITORS LifeArc (GB) 2022-01-19 EP disclosed