SCHEMBL24202

SCHEMBL24202

[CH]1CCc2ccccc2C1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
HTR2C P28335 1/20 0.42
MAOB P27338 3/20 0.37
CYP2A6 P11509 1/20 0.37
PNMT P11086 1/20 0.37
CD44 P16070 1/20 0.37
MAOA P21397 2/20 0.36
DRD2 P14416 1/20 0.36
DRD1 P21728 1/20 0.36
DRD4 P21917 1/20 0.36
DRD5 P21918 1/20 0.36
DRD3 P35462 1/20 0.36
PLAU P00749 1/20 0.34
GRIN2B Q13224 1/20 0.33
CES1 P23141 1/20 0.33
ORAI1 Q96D31 1/20 0.32
ORAI2 Q96SN7 1/20 0.32
ORAI3 Q9BRQ5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4166748 0.85 TSHR (0.56) TSHRHTR2CMAOBCYP2A6PNMT
SCHEMBL2588514 0.84 TSHR (0.57) TSHRHTR2CMAOBCYP2A6PNMT
SCHEMBL4781181 0.82 TSHR (0.62) TSHRHTR2CMAOBCYP2A6PNMT
SCHEMBL23766 0.78
SCHEMBL594989 0.76 TSHR (0.46) TSHRHTR2CMAOBCYP2A6PNMT
SCHEMBL862128 0.73 TSHR (0.56) TSHRHTR2CMAOBCYP2A6PNMT
SCHEMBL862127 0.73 TSHR (0.56) TSHRHTR2CMAOBCYP2A6PNMT
SCHEMBL29351986 0.71
SCHEMBL33555 0.71
SCHEMBL34906 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1904 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117836296-A Pyrazolopyridone compounds 百济神州有限公司 2024-04-05 CN claimed
US-20230348387-A1 NON-LYSOSOMAL GLUCOSYLCERAMIDASE INHIBITORS AND USES THEREOF ALECTOS THERAPEUTICS INC. (CA) 2023-11-02 US claimed
WO-2023148206-A1 MICROBIOCIDAL N-AMIDE DERIVATIVES SYNGENTA CROP PROTECTION AG (CH) 2023-08-10 WO claimed
US-20230174486-A1 NON-LYSOSOMAL GLUCOSYLCERAMIDASE INHIBITORS AND USES THEREOF ALECTOS THERAPEUTICS INC. (CA) 2023-06-08 US claimed
CN-115867534-A Non-lysosomal glucosylceramidase inhibitors and uses thereof 阿勒克图治疗公司 2023-03-28 CN claimed
EP-4146624-A1 NON-LYSOSOMAL GLUCOSYLCERAMIDASE INHIBITORS AND USES THEREOF Alectos Therapeutics Inc. (CA) 2023-03-15 EP claimed
EP-4146623-A1 NON-LYSOSOMAL GLUCOSYLCERAMIDASE INHIBITORS AND USES THEREOF Alectos Therapeutics Inc. (CA) 2023-03-15 EP claimed
CN-115803025-A Non-lysosomal glucosylceramidase inhibitors and uses thereof 阿勒克图治疗公司 2023-03-14 CN claimed
US-20220280527-A1 TRACE AMINE ASSOCIATED RECEPTOR 1 AGONISTS AND PARTIAL AGONISTS FOR PAIN TREATMENT PURDUE PHARMA L.P. (US) 2022-09-08 US claimed
CN-113234194-B Copolymer, primer composition, double-layer system and application of double-layer system in double-layer stripping process 北京科华微电子材料有限公司 2022-08-12 CN claimed
EP-0512352-A2 Substituted carboxylic acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1992-11-11 EP claimed
EP-0213080-B1 HYDROGENATED PYRIDINE DERIVATIVES CIBA-GEIGY AG (CH) 1992-05-20 EP claimed
EP-0304758-B1 N,N'-DIACYLAMINALS BAYER AG (DE) 1991-09-04 EP claimed
US-4987130-A ANTIARRHYTHMIA AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-01-22 US claimed
US-4939160-A Nootropic agents CIBA-GEIGY CORPORATION (US) 1990-07-03 US claimed
EP-0335375-A2 Antihyperlipidemic and antiatherosclerotic compounds and compositions WARNER-LAMBERT COMPANY (US) 1989-10-04 EP claimed
US-4833169-A MEMORY ACTIVATORS CIBA-GEIGY CORPORATION (US) 1989-05-23 US claimed
EP-0286929-A2 Pyrrolidine derivatives, process for their preparation, agents containing them as well as their use HOECHST AKTIENGESELLSCHAFT (DE) 1988-10-19 EP claimed
EP-0213080-A2 Hydrogenated pyridine derivatives CIBA-GEIGY AG (CH) 1987-03-04 EP claimed
US-4152527-A 15-Substituted-ω-pentanorprostaglandins PFIZER INC. (US) 1979-05-01 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230348387-A1 NON-LYSOSOMAL GLUCOSYLCERAMIDASE INHIBITORS AND USES THEREOF GBA1, GBA2, GAA TSHR 3702/4885HTR2C 4681/4885MAOB 1282/4885
US-20220280527-A1 TRACE AMINE ASSOCIATED RECEPTOR 1 AGONISTS AND PARTIAL AGONISTS FOR PAIN TREATMENT TAAR1, TAAR5, OPRL1 TSHR 163/4885HTR2C 208/4885MAOB 454/4885
US-20230174486-A1 NON-LYSOSOMAL GLUCOSYLCERAMIDASE INHIBITORS AND USES THEREOF GBA1, GBA2, GAA TSHR 3702/4885HTR2C 4681/4885MAOB 1282/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.