SCHEMBL24202076

SCHEMBL24202076

C=Nc1ccc2c(c1)CCN2c1ncnc(C)c1/N=C(\C)C=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 4/20 0.34
MKNK2 Q9HBH9 4/20 0.34
EIF4E P06730 3/20 0.34
EGFR P00533 5/20 0.32
CSF1R P07333 1/20 0.32
SRD5A1 P18405 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
HTT P42858 1/20 0.31
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
HSD17B10 Q99714 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
GPR119 Q8TDV5 3/20 0.31
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
PDGFRB P09619 1/20 0.31
TUBA3C P0DPH7 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23761495 0.75 MKNK1 (0.55) MKNK1MKNK2EIF4EEGFRCSF1R
SCHEMBL23761642 0.75 EIF4E (0.35) MKNK1MKNK2EIF4EEGFRCSF1R
SCHEMBL23761308 0.74 MKNK1 (0.48) MKNK1MKNK2EIF4ESRD5A1GPR119
SCHEMBL24201700 0.73 NPC1 (0.41) MKNK1MKNK2EIF4EEGFRCSF1R
SCHEMBL24202017 0.73 NOTUM (0.41) MKNK1MKNK2EIF4EEGFRSRD5A1
SCHEMBL23761492 0.71 MKNK1 (0.45) MKNK1MKNK2EIF4ESRD5A1GPR119
SCHEMBL23761530 0.71 NOTUM (0.40) MKNK1MKNK2EIF4ESRD5A1SMN1; SMN2
SCHEMBL24201658 0.70 SRD5A1 (0.41) MKNK1MKNK2EIF4EEGFRCSF1R
SCHEMBL24201877 0.66 EGFR (0.47) MKNK1MKNK2EGFRCSF1RSRD5A1
SCHEMBL23761414 0.65 SRD5A1 (0.45) MKNK1MKNK2EIF4EEGFRCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3939981-A1 FUSED THIAZOLOPYRIMIDINE DERIVATIVES AS MNKS INHIBITORS LifeArc (GB) 2022-01-19 EP disclosed