SCHEMBL24202017

SCHEMBL24202017

C/C(=N\c1c(C)ncnc1N1CCc2cc(C)ccc21)C(=O)N(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.41
SRD5A1 P18405 2/20 0.38
MKNK1 Q9BUB5 6/20 0.35
MKNK2 Q9HBH9 6/20 0.35
EIF4E P06730 3/20 0.35
KDM4E B2RXH2 2/20 0.34
NPC1 O15118 2/20 0.34
MAPT P10636 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
ALDH1A1 P00352 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
CDK4 P11802 2/20 0.33
CCND1 P24385 2/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23761492 0.90 MKNK1 (0.45) NOTUMSRD5A1MKNK1MKNK2EIF4E
SCHEMBL23761530 0.84 NOTUM (0.40) NOTUMSRD5A1MKNK1MKNK2EIF4E
SCHEMBL24201711 0.84 MKNK1 (0.44) NOTUMSRD5A1MKNK1MKNK2EIF4E
SCHEMBL24202204 0.81 GPR119 (0.37) NOTUMSRD5A1MKNK1MKNK2KDM4E
SCHEMBL24202118 0.80 MKNK1 (0.42) NOTUMSRD5A1MKNK1MKNK2EIF4E
SCHEMBL23761308 0.80 MKNK1 (0.48) NOTUMSRD5A1MKNK1MKNK2EIF4E
SCHEMBL24201720 0.79 KMT2A (0.40) NOTUMSRD5A1MKNK1MKNK2EIF4E
SCHEMBL24201658 0.76 SRD5A1 (0.41) NOTUMSRD5A1MKNK1MKNK2EIF4E
SCHEMBL23761642 0.76 EIF4E (0.35) SRD5A1MKNK1MKNK2EIF4EKDM4E
SCHEMBL23761414 0.74 SRD5A1 (0.45) NOTUMSRD5A1MKNK1MKNK2EIF4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3939981-A1 FUSED THIAZOLOPYRIMIDINE DERIVATIVES AS MNKS INHIBITORS LifeArc (GB) 2022-01-19 EP disclosed