SCHEMBL24206992

SCHEMBL24206992

COc1cc(/C=C/C2CCN(C(=O)OC(C)(C)C)CC2)ccc1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.50
BCHE P06276 1/20 0.49
CYP2D6 P10635 3/20 0.47
ABCB1 P08183 3/20 0.47
CYP1A2 P05177 2/20 0.47
ALOX5 P09917 2/20 0.47
NFKB1 P19838 2/20 0.47
HSD11B1 P28845 2/20 0.47
STAT3 P40763 2/20 0.47
NFKB2 Q00653 2/20 0.47
RELA Q04206 2/20 0.47
NFE2L2 Q16236 2/20 0.47
ALDH1A1 P00352 2/20 0.47
APP P05067 2/20 0.46
KDM4E B2RXH2 2/20 0.46
CA12 O43570 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA3 P07451 2/20 0.46
PKM P14618 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25368200 0.85 STS (0.42) ABCB1ALDH1A1STSMEN1LMNA
SCHEMBL20015271 0.83 ALDH1A1 (0.60) ABCB1ALDH1A1STSMEN1MAPT
SCHEMBL14261793 0.83 ALDH1A1 (0.60) ABCB1ALDH1A1STSMEN1MAPT
SCHEMBL14261792 0.83 GPR119 (0.47) ABCB1ALDH1A1KDM4EPKMMAPT
SCHEMBL4187138 0.82 ALDH1A1 (0.43) ALDH1A1KDM4ELMNAMAPTTHRB
SCHEMBL29673726 0.82 STS (0.43) ABCB1ALDH1A1KDM4ESTSMEN1
SCHEMBL21428573 0.82 STS (0.43) ABCB1ALDH1A1KDM4ESTSMEN1
SCHEMBL4187142 0.82 ALDH1A1 (0.43) ALDH1A1KDM4ELMNAMAPTTHRB
SCHEMBL14261780 0.82 GPR119 (0.48) ABCB1KDM4EPKMSTSMAPT
SCHEMBL14261786 0.80 GPR119 (0.58) ALDH1A1KDM4EMEN1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022012622-A1 DEGRADATION OF (EGFR) BY CONJUGATION OF EGFR INHIBITORS WITH E3 LIGASE LIGAND AND METHODS OF USE BEIGENE, LTD. (KY) 2022-01-20 WO disclosed