SCHEMBL24210652

SCHEMBL24210652

BrCCOc1cccc2c(I)n[nH]c12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.33
FLT3 P36888 1/20 0.33
PLK3 Q9H4B4 1/20 0.33
ITK Q08881 1/20 0.32
HTR1B P28222 3/20 0.32
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
KDM4E B2RXH2 1/20 0.31
HTR1D P28221 1/20 0.31
KCNA3 P22001 1/20 0.30
MEN1 O00255 2/20 0.30
MAPT P10636 2/20 0.30
KMT2A Q03164 2/20 0.30
LMNA P02545 1/20 0.30
MAPK1 P28482 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
HSD17B10 Q99714 1/20 0.30
NPC1 O15118 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30401688 1.00 CHEK1 (0.33) CHEK1FLT3PLK3ITKHTR1B
SCHEMBL17261999 0.85 CHEK1 (0.36) CHEK1FLT3PLK3ITKHTR1B
SCHEMBL5484683 0.76 KDM4E (0.53) CHEK1FLT3PLK3ITKALDH1A1
SCHEMBL30039348 0.76 KDM4E (0.53) CHEK1FLT3PLK3ITKALDH1A1
SCHEMBL15505899 0.72 MCHR1 (0.36) CHEK1FLT3PLK3ITKALDH1A1
SCHEMBL24210984 0.70 NOS1 (0.51) CHEK1FLT3HTR1BALDH1A1HPGD
SCHEMBL30402472 0.70 NOS1 (0.51) CHEK1FLT3HTR1BALDH1A1HPGD
SCHEMBL31127684 0.70 NOS1 (0.41) CHEK1FLT3PLK3KDM4EHSD17B10
SCHEMBL16724769 0.70 NOS1 (0.41) CHEK1FLT3PLK3KDM4EHSD17B10
SCHEMBL25045526 0.69 CHEK1 (0.42) CHEK1FLT3PLK3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113929693-B Nitrogen-containing heterocyclic compound, pharmaceutical composition and application 广州费米子科技有限责任公司 2023-05-09 CN disclosed
WO-2022012534-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION, AND APPLICATIONS 广州费米子科技有限责任公司 2022-01-20 WO disclosed
CN-113929693-A Nitrogen-containing heterocyclic compound, pharmaceutical composition and application 广州费米子科技有限责任公司 2022-01-14 CN disclosed