SCHEMBL2423988

SCHEMBL2423988

Cc1cc(OC(=O)Nc2ccc([N+]3(N4CCC[C@@H]4C)CCCC3)cc2C)on1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HRH3 Q9Y5N1 8/20 0.36
KCNH2 Q12809 2/20 0.36
RAB9A P51151 3/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
TP53 P04637 1/20 0.32
NPC1 O15118 2/20 0.31
CCNE1 P24864 2/20 0.31
CDK2 P24941 2/20 0.31
GSK3B P49841 1/20 0.31
POLB P06746 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2425863 0.85 HRH3 (0.33) MAPTHTTNPSR1HRH3KCNH2
SCHEMBL222647 0.84 KMT2A (0.41) HTTHRH3KCNH2RAB9AKMT2A
SCHEMBL2429279 0.81 HRH3 (0.33) MAPTTSHRHTTNPSR1HRH3
SCHEMBL2421851 0.81 HRH3 (0.35) MAPTHRH3KCNH2RAB9ANPC1
Cyclohexane SCHEMBL2428515 0.80 HRH3 (0.40) HRH3KCNH2RAB9ANPC1CYP3A4
Trifluoroacetic Acid SCHEMBL445482 0.79 HRH3 (0.38) MAPTHTTHRH3KCNH2RAB9A
SCHEMBL223649 0.77 KCNH2 (0.46) MAPTTSHRHTTNPSR1HRH3
SCHEMBL2428638 0.76 HRH3 (0.38) MAPTHRH3KCNH2RAB9ANPC1
SCHEMBL223654 0.76 KMT2A (0.46) HRH3KCNH2RAB9AKMT2AATM
SCHEMBL2422227 0.76 GRM5 (0.40) HRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212283-B1 SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE THEREOF SANOFI SA (FR) 2011-09-21 EP claimed