SCHEMBL2428638

SCHEMBL2428638

CC1(C)CC1(C)C.Cc1cc([N+]2(N3CCC[C@@H]3C)CCCC2)ccc1NC(=O)O

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.38
KCNH2 Q12809 6/20 0.35
CYP3A4 P08684 1/20 0.35
RAB9A P51151 3/20 0.34
NPC1 O15118 2/20 0.34
ITGB3 P05106 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGAV P06756 1/20 0.33
ITGA5 P08648 1/20 0.33
ITGA4 P13612 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclohexane SCHEMBL2428515 0.93 HRH3 (0.40) HRH3KCNH2CYP3A4RAB9ANPC1
SCHEMBL220849 0.86 HRH3 (0.38) HRH3KCNH2CYP3A4RAB9A
SCHEMBL223649 0.84 KCNH2 (0.46) HRH3KCNH2RAB9AMAPT
SCHEMBL223654 0.83 KMT2A (0.46) HRH3KCNH2RAB9A
Trifluoroacetic Acid SCHEMBL222396 0.83 HRH3 (0.35) HRH3KCNH2RAB9A
SCHEMBL222631 0.81 RAB9A (0.47) HRH3CYP3A4RAB9ANPC1MAPT
SCHEMBL2421213 0.81 KMT2A (0.44) HRH3CYP3A4RAB9ANPC1POLB
Trifluoroacetic Acid SCHEMBL444415 0.80 KCNH2 (0.41) HRH3KCNH2RAB9AMAPT
SCHEMBL2423319 0.80 KDM4E (0.56) CYP3A4POLBMAPT
Trifluoroacetic Acid SCHEMBL223098 0.79 KMT2A (0.41) HRH3KCNH2RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2212283-B1 SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE THEREOF SANOFI SA (FR) 2011-09-21 EP claimed