SCHEMBL2424296

SCHEMBL2424296

Nc1ccc(N[C@H]2CCN(C(=O)O)C2)nc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCNK O75909 8/20 0.47
CDK12 Q9NYV4 8/20 0.47
HCAR3 P49019 3/20 0.46
JAK3 P52333 3/20 0.44
CYP3A4 P08684 4/20 0.42
CYP2D6 P10635 4/20 0.42
CYP2C9 P11712 4/20 0.42
HSD11B1 P28845 4/20 0.42
HSD11B2 P80365 1/20 0.42
CCNA2 P20248 2/20 0.41
CDK2 P24941 2/20 0.41
CDK7 P50613 2/20 0.41
CCNH P51946 2/20 0.41
MNAT1 P51948 2/20 0.41
BTK Q06187 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2424299 1.00 CCNK (0.47) CCNKCDK12HCAR3JAK3CYP3A4
SCHEMBL28555866 0.86 CCNK (0.61) CCNKCDK12HCAR3JAK3CCNA2
SCHEMBL28555865 0.86 CCNK (0.61) CCNKCDK12HCAR3JAK3CCNA2
SCHEMBL29240904 0.85 HCAR3 (0.44) CCNKCDK12HCAR3JAK3
SCHEMBL29240908 0.85 HCAR3 (0.44) CCNKCDK12HCAR3JAK3
SCHEMBL28552999 0.85 CCNK (0.60) CCNKCDK12HCAR3JAK3
SCHEMBL28508298 0.85 ALDH1A1 (0.46) CCNKCDK12HCAR3JAK3
SCHEMBL28559024 0.85 CCNK (0.60) CCNKCDK12HCAR3JAK3
SCHEMBL28559025 0.85 CCNK (0.60) CCNKCDK12HCAR3JAK3
SCHEMBL28552998 0.85 CCNK (0.60) CCNKCDK12HCAR3JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367817-A1 INHIBITORS OF DIACYLGLYCEROL ACYLTRANSFERASE Via Pharmaceuticals, Inc. (US) 2011-09-28 EP disclosed
WO-2010065310-A1 INHIBITORS OF DIACYLGLYCEROL ACYLTRANSFERASE VIA PHARMACEUTICALS, INC (US) 2010-06-10 WO disclosed