SCHEMBL24243303

SCHEMBL24243303

Nc1nc(Nc2ccc(N3CCOCC3)cc2)nc2[nH]cc(Cl)c12

nearest known ligand 0.54

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 1/20 0.54
BTK Q06187 1/20 0.54
ITK Q08881 11/20 0.53
TP53 P04637 1/20 0.52
MAPT P10636 1/20 0.52
MAPK1 P28482 1/20 0.52
TTK P33981 1/20 0.49
AURKA O14965 1/20 0.47
AURKB Q96GD4 1/20 0.47
PTGS2 P35354 3/20 0.46
JAK2 O60674 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22513976 0.89 BTK (0.55) JAK3BTKITKTTKAURKA
SCHEMBL24243385 0.84 BTK (0.58) JAK3BTKITKTTKAURKA
SCHEMBL24243330 0.83 JAK3 (0.61) JAK3BTKJAK2
SCHEMBL24243309 0.79 TTK (0.67) JAK3BTKTP53MAPTMAPK1
SCHEMBL17150871 0.78 TP53 (0.53) JAK3TP53MAPTMAPK1TTK
SCHEMBL16344213 0.76 PTGS2 (0.72) TP53MAPTMAPK1AURKAAURKB
SCHEMBL24243290 0.76 JAK3 (0.59) JAK3BTKMAPK1AURKBJAK2
SCHEMBL4417817 0.76 MAPT (0.67) TP53MAPTMAPK1AURKAAURKB
SCHEMBL17908123 0.74 MAPT (0.61) TP53MAPTMAPK1AURKAAURKB
SCHEMBL14694266 0.74 SYK (0.58) TP53MAPTMAPK1AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3950691-A1 PYRAZOLOPYRIMIDINE DERIVATIVES AS KINASE INHIBITOR Daewoong Pharmaceutical Co., Ltd. (KR) 2022-02-09 EP disclosed