SCHEMBL24250199

SCHEMBL24250199

COc1cc2c(O)cccc2cc1C=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 8/20 0.54
TLR2 O60603 1/20 0.50
TLR1 Q15399 1/20 0.50
TLR6 Q9Y2C9 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
ALDH1A1 P00352 6/20 0.49
KDM4E B2RXH2 3/20 0.49
TDP1 Q9NUW8 2/20 0.49
TSHR P16473 1/20 0.49
HPGD P15428 3/20 0.44
HSD17B10 Q99714 2/20 0.44
TRIM24 O15164 2/20 0.42
TRIM33 Q9UPN9 2/20 0.42
TYR P14679 1/20 0.42
AOX1 Q06278 1/20 0.42
ALDH5A1 P51649 1/20 0.42
ABAT P80404 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11230561 0.85 ALDH1A1 (0.55) ERN1TLR2TLR1TLR6ALDH1A1
SCHEMBL18525712 0.84 CYP1A2 (0.44) ERN1TLR2TLR1TLR6CA1
SCHEMBL8501456 0.81 KDM4E (0.52) CA1CA2ALDH1A1KDM4ETSHR
SCHEMBL11229197 0.81 ERN1 (0.54) ERN1TLR2TLR1TLR6CA1
SCHEMBL1298117 0.80 GRIN2D (0.53) ERN1CA1CA2TRIM24TRIM33
SCHEMBL4935526 0.79 ALDH1A1 (0.53) ERN1TLR2TLR1TLR6ALDH1A1
SCHEMBL4059355 0.78 ALDH1A1 (0.61) ERN1TLR2TLR1TLR6ALDH1A1
SCHEMBL8955962 0.76 KDM4E (0.56) CA1CA2ALDH1A1KDM4ETSHR
SCHEMBL29620158 0.75 ALDH1A1 (0.77) CA1CA2ALDH1A1KDM4EHPGD
SCHEMBL8206713 0.75 ALDH1A1 (0.77) CA1CA2ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3536685-B1 BICYCLIC-FUSED HETEROARYL OR ARYL COMPOUNDS AND THEIR USE AS IRAK4 INHIBITORS PFIZER (US) 2022-02-16 EP disclosed