SCHEMBL2425128

SCHEMBL2425128

CC(C)(C)c1ccc(-c2ccc3ccccc3n2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 10/20 0.61
RAB9A P51151 10/20 0.61
MEN1 O00255 3/20 0.61
KMT2A Q03164 3/20 0.61
AR P10275 2/20 0.61
KDM4E B2RXH2 7/20 0.60
SMN1; SMN2 Q16637 6/20 0.60
ALDH1A1 P00352 6/20 0.60
NFKB1 P19838 2/20 0.60
NFKB2 Q00653 2/20 0.60
RELA Q04206 2/20 0.60
MAPT P10636 6/20 0.59
HSD17B10 Q99714 3/20 0.59
CYP3A4 P08684 2/20 0.59
TP53 P04637 2/20 0.59
PKM P14618 2/20 0.59
HPGD P15428 2/20 0.59
GMNN O75496 1/20 0.59
THPO P40225 1/20 0.59
BLM P54132 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30847671 1.00 NPC1 (0.61) NPC1RAB9AMEN1KMT2AAR
SCHEMBL14278925 0.86 RAB9A (0.61) NPC1RAB9AMEN1KMT2AAR
SCHEMBL28898945 0.85 NPC1 (0.46) NPC1RAB9AMEN1KMT2AAR
SCHEMBL12112870 0.84 RAB9A (0.80) NPC1RAB9AMEN1KMT2AAR
SCHEMBL20089432 0.84 NPC1 (0.51) NPC1RAB9AMEN1KMT2AAR
SCHEMBL18858303 0.84 RAB9A (0.51) NPC1RAB9AMEN1KMT2AAR
SCHEMBL17413737 0.83 RAB9A (0.47) NPC1RAB9AMEN1KMT2AAR
SCHEMBL29544777 0.82 NPC1 (0.62) NPC1RAB9AMEN1KMT2AAR
SCHEMBL22734790 0.82 NPC1 (0.62) NPC1RAB9AMEN1KMT2AAR
SCHEMBL16021662 0.82 ESR1 (0.51) NPC1RAB9AMEN1KMT2AAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104910079-B The method that toluene and derivative oxidation one kettle way prepare 4 (3H) Quinazol derivatives 同济大学 2017-08-25 CN disclosed
US-20140378685-A1 PREPARATION OF HETEROLEPTIC METAL COMPLEXES SOLVAY SA (BE) 2014-12-25 US disclosed
US-8680760-B2 Beta-diketone ancillary ligands and their metal complexes used in organic optoelectronic devices NATIONAL TSING HUA UNIVERSITY (TW) 2014-03-25 US disclosed
US-20130331577-A1 PREPARATION OF A FAC-ISOMER FOR A TRIS HOMOLEPTIC METAL COMPLEX SOLVAY SA 2013-12-12 US disclosed
EP-2665735-A1 PREPARATION OF A FAC-ISOMER FOR A TRIS HOMOLEPTIC METAL COMPLEX SOLVAY SA (BE) 2013-11-27 EP disclosed
CN-103298822-A Preparation of a fac-isomer for a tris homoleptic metal complex SOLVAY 2013-09-11 CN disclosed
WO-2013098189-A1 PREPARATION OF HETEROLEPTIC METAL COMPLEXES SOLVAY SA (BE) 2013-07-04 WO disclosed
EP-1902076-B1 LIGHT EMITTING POLYMER MATERIAL, ORGANIC ELECTROLUMINESCENCE DEVICE AND DISPLAY DEVICE COMPRISING LIGHT EMITTING POLYMER MATERIAL SHOWA DENKO KK (JP) 2012-11-21 EP disclosed
WO-2012084219-A1 PREPARATION OF A FAC-ISOMER FOR A TRIS HOMOLEPTIC METAL COMPLEX SOLVAY SA (BE) 2012-06-28 WO disclosed
US-8025987-B2 Light emitting polymer material, organic electroluminescence device and display device comprising light emitting polymer material SHOWA DENKO K.K. (JP) 2011-09-27 US disclosed
US-20100270915-A1 Beta-Diketone Ancillary Ligands and Their Metal Complexes Used in Organic Optoelectronic Devices NATIONAL TSING HUA UNIVERSITY (TW) 2010-10-28 US disclosed
US-20100270915-A1 Beta-Diketone Ancillary Ligands and Their Metal Complexes Used in Organic Optoelectronic Devices NATIONAL TSING HUA UNIVERSITY (TW) 2010-10-28 US disclosed
US-20090096353-A1 LIGHT EMITTING POLYMER MATERIAL, ORGANIC ELECTROLUMINESCENCE DEVICE AND DISPLAY DEVICE COMPRISING LIGHT EMITTING POLYMER MATERIAL SHOWA DENKO K.K. (JP) 2009-04-16 US disclosed
EP-1902076-A1 LIGHT EMITTING POLYMER MATERIAL, ORGANIC ELECTROLUMINESCENCE DEVICE AND DISPLAY DEVICE COMPRISING LIGHT EMITTING POLYMER MATERIAL Showa Dendo K.K. (JP) 2008-03-26 EP disclosed
WO-2006135076-A1 LIGHT EMITTING POLYMER MATERIAL, ORGANIC ELECTROLUMINESCENCE DEVICE AND DISPLAY DEVICE COMPRISING LIGHT EMITTING POLYMER MATERIAL SHOWA DENKO K.K. (JP) 2006-12-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100270915-A1 Beta-Diketone Ancillary Ligands and Their Metal Complexes Used in Organic Optoelectronic Devices PBK, DEK, OSTC NPC1 4443/4885RAB9A 4435/4885MEN1 4347/4885
US-20130331577-A1 PREPARATION OF A FAC-ISOMER FOR A TRIS HOMOLEPTIC METAL COMPLEX FHIT, AP2M1, AP1M1 NPC1 1803/4885RAB9A 2336/4885MEN1 674/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.