SCHEMBL24251672

SCHEMBL24251672

CC1(C)CNc2cccnc2O1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OTUD7B Q6GQQ9 2/20 0.37
AKR1B1 P15121 1/20 0.34
NPC1 O15118 1/20 0.33
GSK3B P49841 1/20 0.33
CYP1A2 P05177 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
MAPT P10636 1/20 0.31
HTT P42858 1/20 0.31
BLM P54132 1/20 0.31
KMT2A Q03164 1/20 0.31
HIF1A Q16665 1/20 0.31
SLC6A2 P23975 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNA7 P36544 1/20 0.31
CHRNA4 P43681 1/20 0.31
HTR3A P46098 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31318500 0.79 OTUD7B (0.40) OTUD7BAKR1B1CYP1A2SMN1; SMN2LMNA
SCHEMBL23175233 0.77 KDM4E (0.44) AKR1B1NPC1GSK3BCYP1A2SMN1; SMN2
SCHEMBL18321939 0.75 CHRNB2 (0.37) NPC1CHRNB2CHRNA7CHRNA4HTR3A
SCHEMBL20269773 0.73 NPC1 (0.30) NPC1
Hydrochloric Acid SCHEMBL29404790 0.73 CHRNB2 (0.36) NPC1MAPTCHRNB2CHRNA7CHRNA4
SCHEMBL30303079 0.72 GAA (0.40) MEN1MAPTKMT2A
SCHEMBL1555141 0.72 GAA (0.40) MEN1MAPTKMT2A
SCHEMBL3109662 0.71 NPC1 (0.49) NPC1GSK3BCYP1A2SMN1; SMN2MEN1
SCHEMBL20290300 0.71 CA12 (0.33) AKR1B1NPC1SMN1; SMN2MEN1LMNA
SCHEMBL31306088 0.71 CA12 (0.33) AKR1B1NPC1SMN1; SMN2MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115836064-B Triazine derivative with EGFR (epidermal growth factor receptor) inhibition activity as well as preparation method and application thereof 上海和誉生物医药科技有限公司 2024-08-27 CN disclosed
CN-115836064-A Triazine derivative with EGFR (epidermal growth factor receptor) inhibitory activity and preparation method and application thereof 上海和誉生物医药科技有限公司 2023-03-21 CN disclosed
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed
WO-2022033455-A1 TRIAZINE DERIVATIVE HAVING EGFR INHIBITORY ACTIVITY, PREPARATION METHOD THEREFOR AND USE THEREOF 上海和誉生物医药科技有限公司 2022-02-17 WO disclosed