SCHEMBL2425312

SCHEMBL2425312

CCOC(=O)C(Cc1cccc(Cl)c1)C(=O)C(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.49
MAPK1 P28482 3/20 0.47
MAPT P10636 1/20 0.47
MMP8 P22894 1/20 0.47
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
ALDH1A1 P00352 3/20 0.45
TP53 P04637 1/20 0.45
PPARG P37231 1/20 0.44
PPARA Q07869 1/20 0.44
KMT2A Q03164 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
TSHR P16473 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MEN1 O00255 2/20 0.42
LMNA P02545 2/20 0.42
HPGD P15428 2/20 0.42
TRPV1 Q8NER1 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2422171 0.90 MMP8 (0.52) PNMTMAPK1MAPTMMP8PDE3B
SCHEMBL10544621 0.87 MMP8 (0.54) PNMTMAPK1MAPTMMP8PDE3B
SCHEMBL2422785 0.86 MMP8 (0.49) PNMTMAPK1MAPTMMP8PDE3B
SCHEMBL15261865 0.86 MMP8 (0.41) MAPK1MAPTMMP8ALDH1A1TP53
SCHEMBL901770 0.84 MMP8 (0.47) PNMTMAPK1MAPTMMP8PDE3B
SCHEMBL5751162 0.83 PNMT (0.54) PNMTMAPTALDH1A1PPARGPPARA
SCHEMBL2425273 0.83 MMP8 (0.46) PNMTMAPK1MAPTMMP8PDE3B
SCHEMBL15261621 0.82 SMN1; SMN2 (0.51) PNMTMAPK1MAPTMMP8ALDH1A1
SCHEMBL2422444 0.82 PNMT (0.44) PNMTMAPK1MAPTMMP8PDE3B
SCHEMBL2428821 0.82 MDM2 (0.51) PNMTMAPK1MAPTMMP8ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011114148-A1 4H- [1, 2, 4] TRIAZOLO [5, 1 -B] PYRIMIDIN-7 -ONE DERIVATIVES AS CCR2B RECEPTOR ANTAGONISTS ASTRAZENECA AB (SE) 2011-09-22 WO disclosed