SCHEMBL24257042

SCHEMBL24257042

CC(C)(O)CCNCc1cccc(Br)c1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.57
CYP2D6 P10635 2/20 0.57
CYP2C19 P33261 2/20 0.57
TAAR1 Q96RJ0 2/20 0.46
KDM4E B2RXH2 1/20 0.42
MTOR P42345 1/20 0.42
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
CARM1 Q86X55 1/20 0.40
PRMT6 Q96LA8 1/20 0.40
RIPK1 Q13546 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL29132456 0.94 CYP1A2 (0.52) CYP1A2CYP2D6CYP2C19TAAR1KDM4E
SCHEMBL10547018 0.80 KMT2A (0.59) KDM4ESIGMAR1MEN1KMT2A
SCHEMBL29132455 0.80 CYP1A2 (0.52) CYP1A2CYP2D6CYP2C19TAAR1KDM4E
SCHEMBL6183546 0.78 CYP1A2 (0.76) CYP1A2CYP2D6CYP2C19TAAR1KDM4E
SCHEMBL16619429 0.78 CYP1A2 (0.61) CYP1A2CYP2D6CYP2C19TAAR1KDM4E
SCHEMBL1420648 0.77 CYP1A2 (0.62) CYP1A2CYP2D6CYP2C19TAAR1KDM4E
SCHEMBL23682794 0.77 CYP1A2 (0.64) CYP1A2CYP2D6CYP2C19TAAR1SIGMAR1
SCHEMBL19633152 0.76 CYP1A2 (0.88) CYP1A2CYP2D6CYP2C19TAAR1HTR2A
SCHEMBL6292536 0.76 TAAR1 (0.50) CYP1A2CYP2D6CYP2C19TAAR1RIPK1
SCHEMBL5275606 0.75 CYP1A2 (0.66) CYP1A2CYP2D6CYP2C19TAAR1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116829540-A Condensed nitrogen heterocycles as sigma ligand compounds and uses thereof 密涅瓦神经科学有限公司 2023-09-29 CN disclosed
WO-2022036080-A1 CONDENSED AZACYCLES AS SIGMA LIGAND COMPOUNDS AND USES THEREOF MINERVA NEUROSCIENCES, INC. (US) 2022-02-17 WO disclosed