SCHEMBL24258265

SCHEMBL24258265

CSN1CC2CC2(CNc2ncnc(N(Cc3ccc(C(F)(F)F)cc3)C3CC3)c2F)C1

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.33
GRIN2B Q13224 4/20 0.32
CYP2D6 P10635 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17501181 0.85 RORC (0.34) RORCGRIN2B
SCHEMBL24258253 0.78 GRIN2B (0.36) GRIN2BCYP2D6KCNH2
SCHEMBL24258278 0.78 GRIN2B (0.35) RORCGRIN2BCYP2D6KCNH2
SCHEMBL23545651 0.76 IRAK4 (0.37) RORCGRIN2BCYP2D6KCNH2
SCHEMBL24258279 0.76 CACNA1B (0.33) RORCGRIN2B
SCHEMBL25436999 0.76 SLC6A2 (0.37) RORCGRIN2BCYP2D6KCNH2
SCHEMBL19640409 0.76 CSF1R (0.36) RORC
SCHEMBL19640732 0.76 RORC (0.34) RORCGRIN2BCYP2D6KCNH2
SCHEMBL17501483 0.75 CYP11B2 (0.39) RORCCYP2D6
SCHEMBL19640536 0.75 RORC (0.35) RORCKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3177612-B1 OPTIONALLY FUSED HETEROCYCLYL-SUBSTITUTED DERIVATIVES OF PYRIMIDINE USEFUL FOR THE TREATMENT OF INFLAMMATORY, METABOLIC, ONCOLOGIC AND AUTOIMMUNE DISEASES NUEVOLUTION AS (DK) 2022-02-23 EP disclosed