SCHEMBL24258306

SCHEMBL24258306

FC(F)c1ccc(CNC2CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.53
RAB9A P51151 1/20 0.53
KMT2A Q03164 1/20 0.53
HRH3 Q9Y5N1 2/20 0.52
POLB P06746 1/20 0.49
GRIN2B Q13224 1/20 0.44
BCHE P06276 2/20 0.42
ACHE P22303 2/20 0.42
BACE1 P56817 2/20 0.42
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10073807 0.83 MEN1 (0.69) MEN1RAB9AKMT2AHRH3POLB
SCHEMBL16980401 0.81 RAB9A (0.53) MEN1RAB9AKMT2AHRH3POLB
SCHEMBL1239998 0.78 BCHE (0.61) MEN1RAB9AKMT2AHRH3POLB
SCHEMBL23545659 0.77 HRH3 (0.50) MEN1RAB9AKMT2AHRH3POLB
SCHEMBL16980536 0.74 POLB (0.59) MEN1RAB9AKMT2AHRH3POLB
SCHEMBL14850003 0.74 SMN1; SMN2 (0.49) MEN1RAB9AKMT2AHRH3POLB
SCHEMBL19650838 0.74 MEN1 (0.42) MEN1RAB9AKMT2AHRH3POLB
SCHEMBL24468257 0.74 CXCR4 (0.39) GRIN2BHDAC1
SCHEMBL3236686 0.74 POLB (0.81) MEN1RAB9AKMT2AHRH3POLB
SCHEMBL2731922 0.74 ACHE (0.61) MEN1RAB9AKMT2AHRH3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3177612-B1 OPTIONALLY FUSED HETEROCYCLYL-SUBSTITUTED DERIVATIVES OF PYRIMIDINE USEFUL FOR THE TREATMENT OF INFLAMMATORY, METABOLIC, ONCOLOGIC AND AUTOIMMUNE DISEASES NUEVOLUTION AS (DK) 2022-02-23 EP disclosed