SCHEMBL24258311

SCHEMBL24258311

CSc1ccc(CN)cn1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 6/20 0.39
HRH3 Q9Y5N1 1/20 0.36
ADRB2 P07550 1/20 0.35
RRM2 P31350 1/20 0.35
ABAT P80404 1/20 0.33
AKT2 P31751 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
CYP2A6 P11509 1/20 0.32
LOX P28300 1/20 0.32
KEAP1 Q14145 2/20 0.32
NFE2L2 Q16236 1/20 0.32
ASIC3 Q9UHC3 1/20 0.32
MAOB P27338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9908277 0.81 L3MBTL1 (0.43) HRH3CYP11B1CYP11B2
SCHEMBL25813170 0.80 PIK3CD (0.44) LOXL2HRH3ADRB2RRM2
SCHEMBL29594784 0.79 POLB (0.36) CYP11B1CYP11B2
SCHEMBL246217 0.79 POLB (0.36) CYP11B1CYP11B2
SCHEMBL247901 0.79 KMT2A (0.36) CYP11B1CYP11B2
SCHEMBL507633 0.79 AOC3 (0.41) LOXL2HRH3ADRB2RRM2ABAT
Hydrochloric Acid SCHEMBL10483859 0.78 KMT2A (0.35) CYP11B1CYP11B2
SCHEMBL10483985 0.77 MC4R (0.41) HRH3
SCHEMBL14903596 0.76 ESR1 (0.41) CYP11B1CYP11B2
SCHEMBL19438349 0.76 ALDH1A1 (0.32) CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3177612-B1 OPTIONALLY FUSED HETEROCYCLYL-SUBSTITUTED DERIVATIVES OF PYRIMIDINE USEFUL FOR THE TREATMENT OF INFLAMMATORY, METABOLIC, ONCOLOGIC AND AUTOIMMUNE DISEASES NUEVOLUTION AS (DK) 2022-02-23 EP disclosed