SCHEMBL2426243

SCHEMBL2426243

C=Cc1cccc(-c2cccc(CO[C@H]3CN(C(=O)[C@@H](NC(=O)OC(C)(C)C)C4CCCCC4)[C@](C)(C(=O)O)C3)c2)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.38
CACNA1B Q00975 2/20 0.37
REN P00797 4/20 0.36
CYP3A4 P08684 1/20 0.35
THRB P10828 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
HTRA1 Q92743 1/20 0.33
ACE P12821 1/20 0.33
KLK5 Q9Y337 1/20 0.32
CMA1 P23946 1/20 0.32
CTRC Q99895 1/20 0.32
NAAA Q02083 1/20 0.32
KLK7 P49862 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2430509 0.89 CACNA1B (0.39) CTSLCACNA1BRENCYP3A4THRB
SCHEMBL2427394 0.85 CYP3A4 (0.34) CYP3A4THRBHSD17B10NAAA
Hydrochloric Acid SCHEMBL2429666 0.85 CYP3A4 (0.36) CYP3A4THRBHSD17B10NAAA
SCHEMBL4294862 0.83 ACE (0.40) CTSLCACNA1BRENCYP3A4THRB
SCHEMBL2426240 0.81 KLK5 (0.40) CTSLCACNA1BRENCYP3A4THRB
SCHEMBL3305393 0.79 CHRM3 (0.35) NAAAKLK7
SCHEMBL4307660 0.72 CACNA1B (0.40) CTSLCACNA1BRENCTSBCTSS
SCHEMBL2426349 0.71 NAAA (0.38) CTSBCTSSCTSKNAAA
SCHEMBL2430508 0.70 CACNA1B (0.41) CTSLCACNA1BRENCYP3A4THRB
SCHEMBL8228152 0.68 CYP3A4 (0.38) CYP3A4THRBHSD17B10NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041159-B1 MACROCYCLIC COMPOUNDS AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2011-09-28 EP disclosed